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4-(2,5-dimethoxyphenyl)-2-{[methyl(propan-2-yl)amino]methyl}phenol
1-[(5-fluoro-2-methylphenyl)methyl]-2-(1H-imidazol-2-yl)-1H-imidazole
1-[(4-methoxyphenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
8-(2-butoxyacetyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(4-{[(furan-2-ylmethyl)(methyl)amino]methyl}phenyl)-5,6-dimethyl-3,4-dihydropyrimidin-4-one
5-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-5-[(2-fluorophenyl)methyl]imidazolidine-2,4-dione
2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl}-7-methoxy-4-methylquinazoline
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(2-oxopyrrolidin-1-yl)acetamide
1-(pyridin-3-yl)-4-(2,4,5-trimethylbenzoyl)piperazine
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(propan-2-yloxy)ethan-1-one
N,N-dimethyl-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]azepan-4-amine
1-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
methyl 3-(4-fluorobenzoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(3-phenylpiperidin-1-yl)acetamide
1-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(ethylamino)-N,4-dimethyl-1,3-thiazole-5-carboxamide
(1S,5S)-3-[(5-cyclopentylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)pyrrolidine-3-carboxamide
1-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4,6-dimethyl-1-[2-({2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]-1,2-dihydropyrimidin-2-one
(3R,9aR)-8-(2-chlorobenzoyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-cyclopropyl-1-[(2-methoxypyridin-3-yl)methyl]-4-methylpyrrolidin-2-one
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-(but-2-yn-1-yl)-N'-(2,4-dimethylphenyl)-N-(furan-2-ylmethyl)propanediamide
1-(2-cyclohexylethyl)-3-({[(2-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
ethyl 2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}acetate
(2R)-2-cyclohexyl-2-hydroxy-N-(1,2-oxazol-3-ylmethyl)acetamide
4-[2-methyl-6-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)pyrimidin-4-yl]morpholine
1-{[5-(1-benzofuran-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,3-dimethylurea
5-phenyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
(2E)-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
9-methoxy-N-methyl-3-[3-(5-methylfuran-2-yl)butyl]-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3S,4S)-1-(2-methoxypyridine-3-carbonyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
2-phenyl-N-[(1S)-1-phenylethyl]-1H-imidazole-4-carboxamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-(2-{4-[2-(pyridin-3-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
2-{3-[1-(dimethylamino)ethyl]phenyl}-1H-1,3-benzodiazole-5-carbonitrile
4-cyclopentanecarbonyl-6-methyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
2-amino-4-(3-chloro-4-hydroxy-5-methoxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
methyl(pyridin-3-ylmethyl){spiro[2.4]heptan-1-ylmethyl}amine
3,5-dimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
5-fluoro-2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3-methyl-1H-indole
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(5-methylfuran-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-methyl-2-oxo-2H-chromen-7-yl)-1H-1,3-benzodiazole-6-carboxylic acid
7-(morpholin-4-ylmethyl)-4-[2-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N3-cycloheptyl-1-cyclopropyl-N5-[(4-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-(1,3-thiazol-2-ylmethyl)acetamide
methyl 9-[(4-fluorophenyl)methoxy]-3-[(2-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate