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2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-5-fluoro-N-methylpyrimidin-4-amine
1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-4-phenylpiperidin-4-ol
1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1-(2,4,6-trimethylpyridin-3-yl)urea
4-(2-methylfuran-3-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
3-{2-[4-(5-methylpyridin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
9-(4-amino-6,7-dimethoxyquinazolin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(3aR,6aR)-2-(2-methoxyethyl)-5-(naphthalene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-phenylethyl)-7-{pyrazolo[1,5-a]pyridine-3-carbonyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
3-[(dimethylamino)methyl]-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
1-(1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
(1s,4s)-4-[4-(3-phenylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
5-oxo-1-[3-(2-phenylacetamido)phenyl]pyrrolidine-3-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(3-phenyl-1,2,4-oxadiazol-5-yl)benzamide
1-methyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}piperidine-3-carboxamide
3-{1-[2-(3-chloro-4-hydroxyphenyl)acetyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3R,4R)-1-(3-fluoro-4-methoxybenzoyl)-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
4-(1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperidin-3-yl)benzoic acid
3-(1H-imidazol-1-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)butanamide
3-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
9-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-3-oxa-9-azaspiro[5.5]undecane
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1λ6-thiomorpholine-1,1-dione
4-oxo-4-phenyl-N-[1-(3-phenylpropyl)piperidin-3-yl]butanamide
N-[(5-chloro-1H-indol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)benzamide
3-cyclopropyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
N-(4-chlorophenyl)-5-{4-hydroxy-1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-(1-methoxybutan-2-yl)piperidine-3-carboxamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-6-(piperidin-4-yl)pyrimidin-4-amine
1-[2-(dimethylamino)ethyl]-4-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)pyrrolidin-2-one
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-benzyl-N,N-dimethyl-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-phenyl-3-[1-(4-phenylbutanoyl)piperidin-4-yl]propanamide
N-benzyl-3-[(4-cyclopentylpiperazin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-(pyrrolidin-3-yl)piperazine
{2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}urea
[4-({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-(1-{7-[2-(2-fluorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)oxolane-3-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
1-(2-fluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2S,4S,5R)-4-[(2-carboxyethyl)carbamoyl]-5-(4-chlorophenyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
N-(1-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
2-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-5-methoxy-4H-pyran-4-one
1-[3-(4-methanesulfonylphenyl)-4-(morpholin-4-yl)phenyl]ethan-1-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-(4-methyl-6-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}pyrimidin-2-yl)phenol
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-indole