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6-methyl-5-{2-oxo-2-[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
N-[2-(3-chlorophenyl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(2S,6S)-1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
8-[(4-fluoro-3-methoxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
1-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-3-methylbutan-1-ol
2-(dimethylamino)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(2-methylphenyl)acetamide
N-[(2R,3R)-2-ethoxy-1'-(1H-indazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(3-fluorophenyl)ethan-1-one
4,4,4-trifluoro-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)butanamide
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-(1,3-benzothiazol-2-ylmethyl)-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)pyridine-3-carboxamide
N-{3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]phenyl}cyclopentanecarboxamide
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
3-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
1-({1-[(6-chloropyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
methyl 3-[2-amino-3-cyano-6-(4-hydroxy-3-methoxyphenyl)pyridin-4-yl]benzoate
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2,3-dihydro-1H-isoindole
(2,1,3-benzoxadiazol-5-ylmethyl)[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
6-methyl-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(2,5-dimethoxyphenyl)methyl]acetamide
1-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
N-(furan-2-ylmethyl)-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(prop-2-yn-1-yl)propanamide
4-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-1-(4-methylphenyl)piperazin-2-one
4-benzyl-2-(hydroxymethyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperazine-1-carboxamide
3-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-3,4-dihydrophthalazine-1-carboxamide
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
1-(4-ethenylphenyl)-3-methyl-3-[2-(methylsulfanyl)ethyl]urea
2-{2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)piperidin-2-one
N4-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N4-methyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(2-oxopyrrolidin-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
9-[(3,5-dichloro-2-hydroxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
6-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-5,6,7,8-tetrahydro-1,6-naphthyridine
2-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
1-{4-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]phenyl}-2-(morpholin-4-yl)ethan-1-ol
3-[(2-methoxyethyl)sulfamoyl]-5-(3-methyl-1H-1,2,4-triazol-1-yl)benzoic acid
ethyl 1-(2-chlorophenyl)-5-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-1H-pyrazole-4-carboxylate
2,5-dimethyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
N,1-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-imidazole-4-sulfonamide
methyl 3-[(3-hydroxy-4-methoxyphenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
1-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-[(3S,4R)-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
2-benzyl-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole