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methyl (2S)-1-{3-[(2,3-difluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}pyrrolidine-2-carboxylate
4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-1-methyl-3-phenyl-1H-pyrazole
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-tert-butyl-5-oxo-N-[3-(pyridin-4-yl)propyl]pyrrolidine-3-carboxamide
3-(1H-imidazol-4-ylmethyl)-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperazin-2-one
2-(2,4-dichlorophenoxy)-N-(oxan-4-yl)acetamide
1,5-dimethyl-3-{[5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-indazole
N3-tert-butyl-N5-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
8-(1-methyl-1H-pyrazole-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
5-methoxy-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-4-oxo-1,4-dihydropyridine-2-carboxamide
5-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridin-3-amine
N-[3-(3,5-dimethylphenoxy)propyl]-3-(3-hydroxy-1,2-oxazol-5-yl)-N-methylpropanamide
3-fluoro-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
2-(4-fluorophenyl)-4-(5-propyl-1,2,4-oxadiazol-3-yl)morpholine
4-fluoro-N-(3-{4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl}phenyl)benzene-1-sulfonamide
N-(3-phenyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-4-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-cyclobutyl-1,3,4-oxadiazol-2-amine
6-methyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)imidazo[1,2-a]pyridine-2-carboxamide
3-[(3R,4S)-1-(2,4-difluorobenzoyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
[(1-ethyl-3-methyl-1H-pyrazol-5-yl)methyl](methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclohex-1-ene-1-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(oxan-4-ylmethyl)benzamide
1-benzyl-8-(furan-3-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-4-(3-hydroxy-3-methylbutyl)-N-(pyridin-3-ylmethyl)benzamide
3-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
N-benzyl-6-(naphthalen-1-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-4-methylpiperazine
N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
5-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(2-methoxyacetamido)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
3-phenyl-N-{1-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
3-({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)-N-(1-phenylethyl)propanamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1,5-dimethyl-2-phenyl-4-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(pyrrolidin-1-yl)ethyl]amine
{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
4-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-[2-({4-benzyl-5-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)ethyl]morpholine
4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[(3-methoxyphenyl)methyl]piperidine-1-carboxamide
N-ethyl-4-hydroxy-2-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyrimidine-5-carboxamide
4-(hydroxymethyl)-1-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperidin-4-ol
[3-(2-phenylethyl)-1-(thiophene-3-carbonyl)piperidin-3-yl]methanol
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-pyrazole-3-carboxamide
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3,3-dimethylbutan-1-one
2-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-{2-[(4-oxopiperidin-1-yl)methyl]phenyl}thiophene-2-carbonitrile
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methoxyphenyl)propanamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-[4-(2,6-dimethoxypyridine-3-carbonyl)piperazin-1-yl]quinazoline
3-{5-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid