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1-(1H-imidazol-2-ylmethyl)-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
2-ethyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}pyrimidine-5-carboxamide
4-[4-(1-acetylpiperidin-4-yl)piperazin-1-yl]-2-[(4-chlorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
8-(dimethyl-1,3-oxazole-5-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{1,3-dimethyl-4-[4-(piperidin-1-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
N-[(3S,4R)-1-(2,6-diaminopyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridine-2-carbonitrile
N3-ethyl-N5-[(2-methylphenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-(7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
N-(thiophen-3-ylmethyl)quinoxaline-6-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-ethylpiperazine
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-(trifluoromethyl)benzamide
3-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propanamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(4-phenylpiperidin-1-yl)acetamide
5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-indazole
1-(2,3-dimethylquinoxalin-6-yl)-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methylurea
1-[(4-ethoxyphenyl)methyl]-4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-(3-{1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
4-[3-cyclopropyl-5-(2,3-dihydro-1,4-benzodioxin-2-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}azepan-4-amine
[(3-ethyl-1,2-oxazol-5-yl)methyl]({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-[3-(trifluoromethyl)benzoyl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
N-(1-cyclopentyl-1H-pyrazol-5-yl)-3-(1-methylcyclopropyl)propanamide
2-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1S)-1-phenylethyl]urea
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-tert-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[1-(2,5-dimethoxyphenyl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
1-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-pyrazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(2-methoxyethyl)(thiophen-2-ylmethyl)amine
5-(azocan-1-yl)-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[3-({[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
2-amino-4-{4-[(dimethylamino)methyl]thiophen-2-yl}-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(morpholin-4-yl)cyclohexane-1-carboxamide
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(1R,9aR)-1-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
(2S)-2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)-3-phenylpropanamide
1-(2-chloropyridine-4-carbonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
5-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
3-[(1-phenylbutyl)carbamoyl]pyridin-1-ium-1-olate
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-({[(dimethylcarbamoyl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
butyl 3-{[(4-fluorophenyl)carbamoyl]methyl}morpholine-4-carboxylate
3-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1λ6-thiane-1,1-dione
5-(1-benzylpiperidin-4-yl)-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione