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3-(3-chlorobenzoyl)-1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidine
5-(2-chloro-4-methoxyphenoxymethyl)-N-ethyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
8-(1,2-oxazole-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-4-methoxyphenol
propyl 2-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane-7-carboxylate
4-methyl-2-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)phenol
methyl 2-[(butan-2-yl)sulfamoyl]-6-(3-phenylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-chloro-6-fluoro-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}benzamide
N4-ethyl-N2-methyl-N2-[2-(oxan-4-yl)ethyl]pyrimidine-2,4-diamine
5-[1-(2-cyclopropylacetyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-indole-6-carboxamide
4-methyl-5-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidin-2-amine
1-[(6-methylpyridin-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-(3-cyclopropyl-5-{[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl)-3-methylpyridine
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
(3R)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3,4,4-trimethylpyrrolidin-3-ol
8-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
[(3-chloro-2,4-difluorophenyl)methyl](methyl)[2-(methylamino)ethyl]amine
(2E)-1-{4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-3-(4-methoxyphenyl)prop-2-en-1-one
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-3-(pyridin-4-yl)propanamide
methyl 3-(7-chloro-2-{[3-(3-methyl-1H-pyrazol-1-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
2-methoxy-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
(1-{[4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-2-yl)methanol
N-[(2S,4R,6S)-2-(2-methylpropyl)-6-(2,3,4-trimethoxyphenyl)oxan-4-yl]acetamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-N,N-diethylpiperidine-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-(3-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
2-(2-hydroxyethyl)-9-(3-methyl-2-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[2-amino-6-(8-methoxy-2-methylquinolin-5-yl)pyrimidin-4-yl]amino}ethan-1-ol
(3S,9aR)-3-(hydroxymethyl)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,3s,6r,8S)-4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
(2R)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxypropanamide
N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylbutanamide
6-[(4-ethylphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{[1-(pyrimidin-2-yl)piperidin-3-yl]amino}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
methyl 5-[(1-methoxypropan-2-yl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(2,6-dimethoxypyridin-3-yl)-1-methyl-1H-indazole
N-[4-(3-methylphenyl)phenyl]-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pyridine-2-carboxamide
3-(but-2-yn-1-yl)-5-[1-(1-phenylcyclopropanecarbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[(3S,4R)-1-(3-fluoro-4-methylbenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
4-{5-[(4-fluoro-3-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-(2,4-difluorophenyl)piperidine-1-carboxamide
methyl({[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl})[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
(3S,4S)-N-(furan-2-ylmethyl)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine