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N-[2-(dimethylamino)ethyl]-2-[2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]acetamide
N-(3-hydroxypropyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
9-hydroxy-2-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
3-methyl-N-{1-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
methyl 3-[(5-methylthiophen-2-yl)methyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-3-methyl-1,2-oxazole
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridin-2-amine
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-[(2-phenylphenyl)methyl]-2,3-dihydropyridazin-3-one
2-{[4-amino-6-(4-methyl-3-phenylpiperazin-1-yl)pyrimidin-2-yl]sulfanyl}-N,N-dimethylacetamide
1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
3-[3-(ethoxymethyl)-5-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
4-(4-chlorophenyl)-1-[4-(2-methylpyridin-4-yl)piperazin-1-yl]butan-1-one
(1S,5R)-3-[4-(piperidin-1-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-(2-methylpropyl)-4-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-dihydropyrimidin-2-one
4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}-N-phenylpiperidine-1-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-{[5-(6-methylpyridazin-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}thiomorpholine
4-(3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
2-[4-(5-{[(3-fluorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]-2-oxoacetamide
2-{5-[(dimethylamino)(3-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-methyl-N-[3-(methylsulfanyl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
(5R)-5-(3,3-diphenylpiperidine-1-carbonyl)pyrrolidin-2-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[1-(thiophen-2-yl)ethyl]benzamide
5-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
1-(2-ethoxypyridine-3-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[2-(4-chlorophenyl)ethyl]-2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]acetamide
6-(3-phenylbutyl)-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
dimethyl[(5-{1-[2-(pyridin-3-yl)ethyl]-1H-imidazol-2-yl}thiophen-3-yl)methyl]amine
methyl 1-{[4-(2,2-diethylcyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
N,N-dimethyl-2-[(1S,5R)-3-(4-methylpyrimidin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
1-[4-({6-chloro-4-[(2-methoxyethyl)amino]quinazolin-2-yl}methyl)piperazin-1-yl]ethan-1-one
3-benzyl-4-(1,5-dimethyl-1H-pyrazole-4-carbonyl)piperazin-2-one
3-{1-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-2-yl}propanoic acid
4-[4-(3-methoxypiperidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
1-benzyl-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-2-one
3-(6-methoxynaphthalene-2-carbonyl)-1-(2-methylfuran-3-carbonyl)piperidine
3-(3-chlorophenyl)-1-(cyclopropylmethyl)-6-(quinoxalin-5-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-{5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}acetic acid
(3aS,6aS)-2-{[5-(methylcarbamoyl)furan-2-yl]methyl}-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-amino-6-(5-methyl-1H-indol-3-yl)pyrazin-2-yl]piperidine-3-carbonitrile
3-(2-chloropyridin-3-yl)-1-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}urea
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]morpholine-2-carboxamide
3-{ethyl[(1-phenyl-1H-pyrazol-5-yl)methyl]amino}-1λ6-thiolane-1,1-dione
N-[2-(3,5-dimethylphenoxy)ethyl]-N,1-dimethyl-5-oxo-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4aS,7aR)-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]cyclopropane-1-carboxamide
1-(benzyloxy)-8-[2-(2-chloro-4-fluorophenyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
2-acetyl-7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N4-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-6-(propan-2-yl)pyrimidine-2,4-diamine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine