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(3aS,6aS)-2-[(prop-2-en-1-yl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
methyl N-{2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}carbamate
3,5-dimethyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
1-(3-chloro-4-methoxybenzoyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(pyridin-4-ylmethyl)propanamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(pyridin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
2-(3-fluorophenyl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
3-({4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)-1-methanesulfonylpiperidine
1-[(2,3-difluorophenyl)methyl]-4-[1-(5-ethyl-1,3-oxazole-4-carbonyl)pyrrolidin-3-yl]piperidine
9-(3-phenylpropanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-methoxyphenyl)-4-[2-(oxan-2-ylmethoxy)acetyl]piperazin-2-one
5-[methyl(2-phenylethyl)amino]-2-[(4-methyl-1,3-thiazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
7-(3-chlorophenyl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S)-2-acetamido-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-(methylsulfanyl)butanamide
4-{[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
3-(2,4-difluorophenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-methoxy-3-(2-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)propan-2-ol
3-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-{1-[1-(2-methoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
2-[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]acetic acid
N-ethyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-(2-methylprop-2-en-1-yl)acetamide
1-tert-butyl-N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
{3-[(3-methylpyrazin-2-yl)methyl]-9-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-(benzylsulfamoyl)piperidine-3-carboxamide
5-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]quinoxaline
2-methyl-4-(4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
(3S,4R)-1-[4-(2-methoxyphenyl)benzoyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-{2-[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
2-(3-methoxypropyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-methyl-N-(pyridin-3-ylmethyl)furan-2-carboxamide
4,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidin-2-amine
1-(2-chlorophenyl)-3-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
3-{[(2,5-dimethylpyrimidin-4-yl)amino]methyl}-2-methoxy-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidin-3-yl}benzoic acid
2-cyclopentyl-N-(2-{5-[(2,3-dihydroxypropyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)acetamide
2-{2-[1-(2-methylquinoline-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-cyclopentyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-ethyl-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-oxazole-4-carboxamide
7-[(4-fluorophenyl)methyl]-2-(5-methyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]-N-(3-hydroxypropyl)acetamide
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2,2-dimethylpropan-1-one
2-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{3-oxo-9-[3-(thiophen-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
4-(cyclopropylmethyl)-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-(carbamoylmethyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}piperidine-3-carboxamide
N-cyclopropyl-N-({4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-5-methylthiophene-2-carboxamide
3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide