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6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,N-dimethylpyrimidin-4-amine
dimethyl[2-(3-{3-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)ethyl]amine
3-({1-[(2-ethylpyrimidin-4-yl)methyl]pyrrolidin-3-yl}methyl)-1-phenylurea
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-methylphenyl)methyl]piperidine-3,5-dicarboxamide
N-benzyl-6-(dimethylamino)-N-[1-hydroxy-3-(1H-imidazol-5-yl)propan-2-yl]pyridine-3-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(3-methylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methyl-1,3-thiazole-4-carboxamide
N-methyl-N-[2-(4-methylphenoxy)ethyl]-2-oxo-1,3-oxazolidine-4-carboxamide
1-cyclohexyl-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
1,3-dimethyl-N-(oxolan-3-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-(1-phenylethyl)benzamide
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
N-benzyl-1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(2-hydroxyethyl)piperidine-4-carboxamide
N,3,5-trimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-benzofuran-2-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-2,5-dimethoxy-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
(4aS,7aR)-1-[2-(dimethylamino)acetyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)(pyrrolidin-1-yl)methyl]pyridine
(1,3-benzothiazol-2-ylmethyl)({[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-cyclohexyl-3-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propanamide
N'1-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}cyclopropane-1,1-dicarboxamide
(1R,3S)-7-(3-fluoro-4-methylbenzoyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
2-methyl-4-{4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
2-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-1-methyl-1H-indole
N-[1-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide
(cyclopropylmethyl)({[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl})propylamine
4-({2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
methyl 4-{[(2S,4S)-2-({2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}carbamoyl)-4-(pyrimidin-2-ylsulfanyl)pyrrolidin-1-yl]methyl}benzoate
3-[(4-fluorophenyl)methyl]-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-5-carboxamide
4-hydroxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(butan-2-yl)-N3-ethyl-N5-[(3-fluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
1-(3,5-difluoropyridine-2-carbonyl)-4-(3-methoxybenzoyl)piperazine
6-methyl-2-{[4-(2-propoxyethyl)piperazin-1-yl]methyl}quinolin-4-ol
2-(1,2-benzoxazol-3-yl)-N-[1-(butan-2-yl)-1H-pyrazol-5-yl]acetamide
7-[(4-fluorophenyl)methyl]-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-[3-(pyrrolidin-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(2-benzyl-1,3-thiazole-4-carbonyl)-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoyl}-1,4-diazepane-1-carbaldehyde
4-{[(3aS,6aS)-3a-carboxy-5-(cyclohexylmethyl)-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
1-cyclohexyl-N-methyl-N-(oxan-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(4-hydroxypiperidin-1-yl)acetamide
1-(4,6-dimethylquinazolin-2-yl)-N-(1-hydroxy-2-methylpropan-2-yl)piperidine-4-carboxamide
2-methyl-7-[3-(pyridin-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aS,8aS)-2-[(3-phenylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-butyl-8-cycloheptyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
7-(3-phenylpropyl)-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane