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2-(2-methoxy-4-methylphenoxymethyl)-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
1-[2-(cyclohexylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-methyl-8-(5-methylthiophene-2-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-({3-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-N-cyclopentyl-2-fluorobenzamide
2-[(2-methylpyrimidin-5-yl)methyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxypyridine-3-carboxamide
[(2,3-dimethoxyphenyl)methyl]({[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl})amine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
6-amino-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]hexan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(1H-pyrazol-1-yl)benzamide
(2S,4R)-N-[2-(3-chlorophenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
N-[(1S)-3-(methylsulfanyl)-1-[1-phenyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]propyl]acetamide
2-(2-hydroxyethyl)-9-[3-(5-methylfuran-2-yl)butyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
1-(3-phenylpropyl)-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
(1S,5R)-6-(2,6-difluorobenzoyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[(3R,4R)-3-hydroxy-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
propan-2-yl 4-chloro-3-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]amino}benzoate
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}benzonitrile
(3R,4R)-4-ethyl-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidine-3,4-diol
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(2-methoxyethyl)-5-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
3-(3-fluorophenyl)-4-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-[4-(4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
2-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,4-dihydroquinolin-4-one
2-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}benzoic acid
N-[(3-chloro-2-methylphenyl)methyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-hydroxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclobutan-1-amine
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2,1,3-benzothiadiazole-4-sulfonamide
(2R,3R,6R)-N-butyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
1-cyclopropanecarbonyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidine-4-carboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
(2R,3R,6R)-3-phenyl-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-ethyl-6-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
N,N-diethyl-1-{1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-(dimethyl-1,3-thiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
2-(2,3-difluorophenoxymethyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
[1-({4-[(2-fluoro-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-2-yl]methanol
1-(5-chloropyridin-2-yl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
1-[7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,2-diphenylethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S,9aS,9bS)-5-(1H-imidazol-2-yl)-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(oxan-4-ylmethyl)piperidine-4-carboxamide
1-[4-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)piperidin-1-yl]ethan-1-one
N-benzyl-3-{[(1,4-dithiepan-6-yl)amino]methyl}-N-methylpyridin-2-amine