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5-(3-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
1-(furan-2-ylmethyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidine-4-carboxamide
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-3-{[4-(propan-2-yl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanamide
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-2-(trifluoromethyl)benzamide
N-ethyl-2-methyl-N-[2-(3-methylphenoxy)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[2-(4-chlorophenyl)ethyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
5-(furan-2-ylmethyl)-5-{3-[3-(2-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}quinoxaline
8-[(3-hydroxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 3,5-dimethyl-4-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)carbamoyl}-1H-pyrrole-2-carboxylate
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
2-(2-{[(2R)-2-methylpiperazin-1-yl]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
4-[7-(5-fluoropyrimidin-2-yl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
2-(4-fluorophenyl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(piperidin-1-yl)ethan-1-one
N-(1-carbamoylcyclopentyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
5-[(1-benzyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
6-[2-(pyrimidin-2-ylsulfanyl)acetyl]-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
5-(3-methoxyphenoxymethyl)-N-[2-(pyridin-3-yloxy)propyl]-1,2-oxazole-3-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
[(1-benzyl-1H-pyrazol-4-yl)methyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
7-[(4-fluorophenyl)methyl]-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
(1R,2R,6S,7S)-4-(2-phenoxybenzoyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-(ethylamino)-N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)pyrimidine-5-carboxamide
N-ethyl-6-oxo-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-(5-aminopentyl)-2-(dimethylamino)-2-(4-methylphenyl)acetamide
(3S,9aR)-3-benzyl-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(3-ethylphenyl)-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-methyl-5-(3-methyl-3-phenylpiperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1-{7-[(9-ethyl-9H-carbazol-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
2-[(6-{4-[1-(morpholin-4-yl)ethyl]phenyl}quinazolin-4-yl)amino]ethan-1-ol
N-{3-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-oxopropyl}methanesulfonamide
(2S)-2-amino-4-[1-(2-chlorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]butanoic acid
5-fluoro-1-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
N-{[1-(1-methylpiperidin-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}cyclopropanamine
(dicyclopropylmethyl)({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)methylamine
N-methyl-1-[2-(1H-pyrazol-1-yl)benzoyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-2-(2-fluorophenyl)ethyl]-N,2-dimethylfuran-3-carboxamide
2-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}-5-methoxyphenol
3-fluoro-4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-[(2R,3R)-2-methoxy-1'-[(3-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
1-[(2-fluorophenyl)methyl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-phenyl-1H-pyrazole-4-carboxamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
2-methyl-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-oxazepane
methyl 5-{[(3,5-difluorophenyl)methyl]amino}-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(4aS,8aR)-6-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one