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N-[3-(2-methoxyphenyl)propyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(4-methylphenyl)methyl]-2-oxa-7-azaspiro[4.5]decane-7-carboxamide
6-methyl-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
1-{2-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-(6-chloropyridin-3-yl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carboxamide
2-[2-(cyclohexylamino)pyrimidin-5-yl]-N-ethyl-N-methylquinoline-4-carboxamide
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-(quinolin-8-yl)urea
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-(1H-pyrazol-4-yl)benzamide
2,8-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}quinoline-4-carboxamide
4-{[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxypropan-1-one
3-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
[(1-{1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
4-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
2-[2-(dimethylamino)pyrimidin-5-yl]-N,N-diethyl-6,8-dimethylquinoline-4-carboxamide
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-imidazole
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
1-benzyl-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-[(1-phenylcyclopentyl)methyl]acetamide
1-{2-[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(7-methoxy-4-methylquinazolin-2-yl)-N-methyl-N-(oxan-2-ylmethyl)piperidine-3-carboxamide
N-[4-(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)phenyl]acetamide
methyl 1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-4-carboxylate
3-phenyl-6-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyridazine
(2R,6R)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
6-methyl-2-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)quinolin-4-ol
5-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2,3-dimethylbenzene-1-sulfonamide
4-[(3-chloro-2-fluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
7-methoxy-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
ethyl 2-[({[2-(azocan-1-yl)pyridin-3-yl]methyl}carbamoyl)amino]acetate
2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-(2,4-dimethylphenyl)acetic acid
2-[5-(2,3-dihydro-1H-inden-1-yl)-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[3-(morpholin-4-yl)propyl]-5-[4-(2-phenylethyl)piperidine-1-carbonyl]piperidin-2-one
2-(ethylamino)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-4-methyl-1,3-thiazole-5-carboxamide
(4aR,8aS)-1-(2-methoxyethyl)-6-[(4-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]-1-(1-propylpiperidin-4-yl)piperidine
2-{4-[(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenoxy}ethan-1-ol
3-[(diethylamino)methyl]-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
4-(dimethyl-1,3-thiazol-5-yl)phenol
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3,5-dimethyl-1H-pyrrole-2-carboxamide
methyl (1R,3S,3aR,6aS)-3-(5-ethylpyridin-2-yl)-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(2R,3R)-2-hydroxy-1'-(pyridin-4-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
3-ethyl-6-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
6-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-5,6-dihydro-1,6-naphthyridin-5-one
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-phenylprop-2-yn-1-one