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(1R,2S,9R)-11-[(1-methyl-1H-imidazol-2-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]formamido}acetic acid
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]thian-4-amine
{[4-(1H-imidazol-1-yl)phenyl]methyl}(1H-imidazol-2-ylmethyl)methylamine
4-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]morpholine
2-(methylamino)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
ethyl 5-(thiophene-3-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
(2S,4S)-4-amino-N-ethyl-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidine-2-carboxamide
3-(3,4-dimethoxybenzoyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
1-tert-butyl-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-oxopyrrolidine-3-carboxamide
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
1-(1,3-benzoxazol-2-ylmethyl)-3-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)urea
1-cyclopentyl-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazin-2-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(1H-1,3-benzodiazol-2-yl)propan-1-one
2-methoxy-2-phenyl-N-{1-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-({7-[2-(2-methoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
(4aR,8aR)-7-(3-chloro-4-methylbenzoyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
3-{1-methyl-5-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
1-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-3-(thiophen-2-yl)propan-1-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)-1H-imidazole
(2E)-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylpent-2-enamide
3-(hydroxymethyl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-ol
2-chloro-5-acetamido-N-(2-phenoxyethyl)benzamide
N-cycloheptyl-3-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]propanamide
3-[(2-fluorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-(2-amino-6-methylpyrimidin-4-yl)-1-methylpiperazin-2-one
1-benzyl-8-[(4-chlorophenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-2-phenyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-imidazole-4-carboxamide
2-acetamido-3-methyl-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
(4-methyl-5-{[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
N-(2,1,3-benzothiadiazol-4-yl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1-(4-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
5-chloro-3-[2-(3-hydroxypiperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
8-(2H-1,3-benzodioxole-5-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide
ethyl 4-[4-(1H-pyrazol-3-yl)benzamido]piperidine-1-carboxylate
(1S,5R)-6-benzyl-3-[2-(3-methoxyphenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
3-(3-amino-1H-indazol-1-yl)-5-(azepane-1-sulfonyl)benzoic acid
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]acetamide
2,7-dimethyl-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N,6-dimethylpyrimidin-2-amine
2-(1,3-benzothiazol-2-ylmethyl)-4-[3-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)azepane
N-methyl-3-[methyl({4-[(2-methylprop-2-en-1-yl)oxy]phenyl}carbamoyl)amino]butanamide
4-ethyl-3-{[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one