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N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
(4S)-3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
1-cyclopentyl-N-[2-(4-fluorophenoxy)ethyl]-6-oxopiperidine-3-carboxamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(3-phenyl-1H-1,2,4-triazol-5-yl)acetamide
1,3-dimethyl-4-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)piperazin-2-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-butyl-N-(furan-2-ylmethyl)propanamide
N-(4-methoxyphenyl)-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-cyclopropyl-5-(2-methoxy-4-methylphenoxymethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
methyl 1-methyl-4-[3-(1H-pyrazol-1-yl)phenyl]-1H-pyrazole-5-carboxylate
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,4-diazepan-2-one
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,N-dimethyl-2-{4-[3-(2-oxoimidazolidin-1-yl)benzoyl]morpholin-3-yl}acetamide
2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyridine-4-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(2-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl][(1-methyl-1H-imidazol-2-yl)methyl]amine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(1-ethylpyrrolidin-2-yl)methyl]benzamide
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methyl-3-phenyl-1H-pyrazole-5-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amine
(4S)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-3,3,4-trimethylpiperidin-4-ol
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
6-{4-[(1-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-9H-purine
2-(2-{[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,N-diethyl-5-methyl-1H-pyrazole-4-carboxamide
N-{3-[4-(2-hydroxyethyl)piperazine-1-carbonyl]phenyl}oxolane-2-carboxamide
2-({6-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
1-(3-phenylpropyl)-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]piperidin-2-one
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
ethyl 4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
1-methyl-4-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}piperazine
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-N-(furan-2-ylmethyl)piperidine-4-carboxamide
1-(3-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(1-cyclopropanecarbonylpiperidin-4-yl)-4-(2,3-dihydro-1H-inden-2-yl)piperazine
4-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
(1R,9aR)-1-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amino}methyl)-octahydro-1H-quinolizin-1-ol
1-[(4aR,8aS)-6-(2-phenylethyl)-decahydro-1,6-naphthyridin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
5-[(1-carbamoylcyclopentyl)amino]-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-(3-methoxybutyl)-1-[2-(3-methoxyphenyl)phenyl]urea
4-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2-(3,4-dichlorophenyl)morpholine
1-(4-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
[(2S,6S)-11-methoxy-4-[(5-methylthiophen-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-{2-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
N-[(3S,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
(3R,4R)-1-(1,4-dithiepan-6-yl)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
1-(2-acetylbenzoyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
(3S,4R)-1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid