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N-(2-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
5-oxo-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidine
5-hydroxy-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}pyrazine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methylpyrido[2,3-d]pyrimidin-4-amine
3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
6-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-N-[4-(1H-pyrazol-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
3,5-dimethyl-1-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}propyl)-1H-pyrazole
1-[1-(4-methanesulfonylphenyl)ethyl]-3-(2,4,6-trimethylpyridin-3-yl)urea
3-acetamido-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)propanamide
2-({[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)phenol
methyl 1-(2-methoxyethyl)-3-(2-phenylacetamido)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)oxolane-2-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(1,3-thiazol-2-yl)pyrrolidin-3-amine
2-(dimethylamino)-8-[(6-methoxypyridin-3-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[(dimethylamino)methyl]-1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-3-ol
{3-[(dimethylamino)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}methanol
3-methoxy-N-methyl-N-{[3-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
5-ethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 7-oxo-9-(pyridin-4-ylmethoxy)-3-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{methyl[5-(2-methylphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}propane-1,2-diol
[1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[2-(morpholin-4-yl)butyl]amine
N-(3-chloro-4-fluorophenyl)-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}propanamide
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(2-fluorophenyl)methyl](2-methoxyethyl)amine
3-acetamido-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
2-(6-ethyl-2-methylquinoline-4-carbonyl)-1,2-oxazolidin-4-ol
N-[2-(1H-imidazol-2-yl)ethyl]-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-2-methylpyridine
methyl 7-oxo-9-(pyridin-4-ylmethoxy)-3-{[4-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[1-(4-methoxyphenyl)ethyl]methylamine
1-[(2-fluoro-5-methoxyphenyl)methyl]-2-phenylazetidine
2-methoxy-4-[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]phenol
2-[(1E)-3,3-dimethylbut-1-en-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
N3-(1-benzylpiperidin-4-yl)-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[(2,1,3-benzoxadiazol-5-ylmethyl)(thiophen-2-ylmethyl)amino]butan-1-ol
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-2-hydroxybenzamide
1-cyclohexyl-3-(4-phenylpiperidine-1-carbonyl)-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
1-[1-(2-carbamoylethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-phenylbutanamide
2-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
8-(6-chloroquinolin-2-yl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
N-(4-methylphenyl)-3-oxo-3-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]propanamide
6-cyclopropyl-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methylpyrimidin-4-amine
1-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-6-azaspiro[2.5]octane
2-{4-[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
[1-(1-phenylpiperidin-4-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol