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methyl 2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}pentanoate
2-[cyclopentyl(methyl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
14-(6-methoxypyridin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-methyl-6-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,3-benzothiazol-2-amine
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1-benzothiophene-5-carboxamide
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pent-4-ynamide
7-methyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]thieno[3,2-d]pyrimidin-4-amine
2-(furan-2-carbonyl)-1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-[2-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-one
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}urea
5-{[(3-fluoro-4-methylphenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(5-methyl-1,2-oxazol-3-yl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
2-{1-[(3,4-difluorophenyl)methyl]-4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}piperazin-2-yl}ethan-1-ol
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)oxolane-3-carboxamide
N-{1-oxaspiro[4.5]decan-3-yl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-6-ol
1-(difluoromethyl)-5-methyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazole
5-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1,3,4-oxadiazol-2-amine
N-(1-{4-[4-(4-fluorophenoxy)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2-methoxyacetamide
N-[(2R,3R)-2-ethoxy-1'-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-butyl-3-methyl-4-oxo-N-(thiophen-3-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
4-(4-methoxyphenyl)-4-oxo-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
pyridin-2-yl(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidin-4-yl)methanol
N-methyl-N-(2-phenyl-1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-cyclobutyl-N,1-dimethyl-7-(oxolane-2-amido)-N-(thiophen-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
ethyl 1-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]piperidine-2-carboxylate
3-({2-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(4-methoxyquinazolin-6-yl)benzamide
1-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-4-phenylpiperidine-4-carbonitrile
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-[3-(phenylsulfanyl)propyl]acetamide
3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
({2-[(2-chlorophenyl)methoxy]-7-fluoroquinolin-3-yl}methyl)({imidazo[2,1-b][1,3]thiazol-6-ylmethyl})amine
2-(4-methoxyphenyl)-N-({1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}methyl)acetamide
1-[4-(1,3-thiazol-4-yl)phenyl]-N-(thiophen-3-ylmethyl)piperidin-4-amine
1-[(3-chlorophenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-3-carboxamide
2-[({5-[1-(2,2-dimethylpropyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
N-(2H-1,3-benzodioxol-5-yl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-amine
N-{2-[4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)morpholin-2-yl]ethyl}acetamide
3,5-dimethyl-1-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]-1H-pyrazole
(3aR,6aS)-5-(5-ethylthiophene-3-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
dimethyl[(5-{1-[1-(pyridin-2-yl)propyl]-1H-1,2,3-triazol-4-yl}thiophen-3-yl)methyl]amine