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2-cyclobutyl-5-(2-methoxyacetamido)-N,1-dimethyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
3-{[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}-N-methylbenzamide
[9-(cyclopropylmethyl)-3-[(4-fluoro-3-methoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
(4aR,7aS)-1-(2-hydroxyethyl)-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[(2-ethoxyphenyl)methyl]-4-(isoquinolin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
5-(methoxymethyl)-N-(4-{5-methyl-4-[(phenylformamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-2-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-5-methyl-2,1,3-benzothiadiazole-4-sulfonamide
4-methyl-1-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidine-4-carbonitrile
6-{1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]piperidin-3-yl}-2-methyl-3,4-dihydropyrimidin-4-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
3-[3-(aminomethyl)phenyl]-1-ethyl-1-[2-(3-ethylphenoxy)ethyl]urea
{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
6-(2,5-dimethylfuran-3-yl)-N-(2-methoxyethyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{5-[(4-{4-ethyl-1-[2-(4-methoxyphenyl)ethyl]-2,5-dioxoimidazolidin-4-yl}piperidin-1-yl)methyl]thiophen-2-yl}acetamide
3-[(1-cyclopentanecarbonylpiperidin-4-yl)methyl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-cyclopentyl-4-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)piperazin-2-one
1-{3-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-3-oxopropyl}azepan-2-one
5-methyl-5-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
ethyl 4-[3-({[2-(2-fluorophenyl)ethyl]amino}methyl)-6,7-dimethoxyquinolin-2-yl]piperazine-1-carboxylate
3-{4-[(4-fluoro-3-methoxyphenyl)methyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
N-[(3S,4R)-1-phenylmethanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2,3-dimethyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]quinoxaline-6-carboxamide
2-(2-{[4-(ethylamino)pyrimidin-2-yl]amino}ethyl)-1,2-dihydrophthalazin-1-one
1-(3-hydroxyphenyl)-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]propanamide
N-[(3-chlorophenyl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[(2-chlorophenyl)methyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(4S,4aS,8aR)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
N-[1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
N-(2-methoxyphenyl)-3-[(6-methoxypyrimidin-4-yl)amino]propanamide
(2S,4S)-4-benzamido-N-ethyl-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
(1R,3S)-7-(5-chloropyridine-3-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
2-(3-methoxypropyl)-9-{[3-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)acetate
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-5-methylthiophene-2-carboxamide
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-(2-methoxyethyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
5-propyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}benzonitrile
2-cyclopentyl-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-propylpyridine
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
4-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]morpholine
5-cyclopropanecarbonyl-1'-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl (2S)-2-{[2-(4-methoxybenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl]formamido}-2-phenylacetate
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
(2E)-1-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(thiophen-2-yl)prop-2-en-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide