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2-methyl-5-(4-{2-[(2-methylphenyl)sulfanyl]acetyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
3-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
(3R,4S)-4-(3-methoxyphenyl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidin-3-amine
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-2-methoxybenzamide
4-(2-fluorophenoxy)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
[4-({4-[methyl(phenyl)amino]phenyl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl](pyridin-2-yl)methanol
2-{[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-(azepane-4-carbonyl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
4-[(4-fluorophenyl)sulfanyl]-1-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine
N-[1-(1-cyclooctylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
N-benzyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-(oxolan-2-ylmethyl)acetamide
[(3R,4R)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
2-oxo-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1,2-dihydroquinoline-4-carboxamide
2-(hydroxymethyl)-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-1,3-benzodiazole-5-carboxamide
methyl (2S,4S)-1-[(4-hydroxy-3-methoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
N-cyclopentyl-4-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-4-oxobutanamide
2-(3-methyl-3-phenylpiperidine-1-carbonyl)thiophene-3-sulfonamide
1-(cyclohexyloxy)-3-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)propan-2-ol
ethyl 4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
ethyl 4-oxo-5-phenoxy-1-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3-carboxylate
6-methyl-2-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}pyridine-3-carboxamide
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}urea
2-[3-(methanesulfonylmethyl)piperidin-1-yl]pyrimidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4,7-dimethylquinazolin-2-yl)piperidine-3-carboxamide
4-oxo-5-phenoxy-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,4-dihydropyridine-3-carboxylic acid
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-(piperidin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
6-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]-4-(2-methylpropyl)-1-(propan-2-yl)-1,4-diazepan-2-one
N-[(2R,3R)-1'-[(4-fluoro-3-methoxyphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
3-(thiophene-2-carbonyl)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
(2S,4R)-4-amino-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
4-phenyl-3-[1-(pyrimidin-2-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 8-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl 2-{5-[1-(2,3-dihydro-1-benzofuran-7-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
N-(1-benzyl-3-methyl-1H-pyrazol-5-yl)thiomorpholine-4-carboxamide
3-benzyl-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
2-[(4-methoxyphenyl)methyl]-4-(thiophene-3-sulfonyl)morpholine
methyl 5-({[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamoyl}amino)-2-chlorobenzoate
1-{4-oxo-4-[2-(2-phenylethyl)morpholin-4-yl]butyl}pyrrolidin-2-one
N-(cyclohexylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2-(3-phenylpropyl)morpholine
2-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
(1S,5R)-3-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole