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N6-benzyl-N5-methyl-N5-[2-(oxan-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
ethyl 3-{[(3aS,6aR)-2-oxo-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carbonyl]amino}propanoate
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-methylpyridine-3-carboxamide
7-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2,3,4-tetrahydroquinoxalin-2-one
3-methyl-1-propyl-4-[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-ethyl-5-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)-1-[(3,4,5-trimethoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-{3-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
4-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
N-[1-(thiophen-3-yl)propan-2-yl]quinoxaline-6-carboxamide
(1R,6S)-9-methyl-3-(2-methyl-5-propylpyrimidin-4-yl)-3,9-diazabicyclo[4.2.1]nonane
1-(2-{[4-methyl-7-(methylsulfanyl)quinolin-2-yl]amino}ethyl)piperidine-3-carboxamide
4-methyl-3-{6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzene-1-sulfonamide
N-({7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenoxyacetamide
2-[2-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)phenoxy]propanoic acid
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-[2-(1-cyclopentylpiperidin-4-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
1-ethyl-4-{[methyl({[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyrrolidin-2-one
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(1-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
3-(3-chlorobenzoyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
1-[2-(4-methoxyphenyl)ethyl]-4-[(1-methylpiperidin-4-yl)amino]pyrrolidin-2-one
({3-[1-(dimethylamino)ethyl]phenyl}methyl)(methyl)[(3-methylpyridin-2-yl)methyl]amine
N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-3,5-dimethyl-1-benzofuran-2-carboxamide
(4aS,8aR)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
2-[4-(cyclopropylmethyl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(3-chlorophenyl)-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
3-{2-[5-(2,3-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
5-ethyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methylpyrimidin-4-amine
methyl (2S,4R)-1-[(2-methoxyphenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
N-[(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]acetamide
N-(2,3-dihydro-1H-inden-1-yl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-chloro-N-{3-[(3-methoxyphenyl)carbamoyl]phenyl}-1-methyl-1H-pyrazole-3-carboxamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(thiophen-3-ylmethyl)propanamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-(prop-2-en-1-ylsulfanyl)ethan-1-one
N-[(5-fluoro-2-methylphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-{4-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-(methylsulfanyl)pyridine
5-{[1-(3-chloro-4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,3-thiazol-2-amine
(2S)-2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2-phenylethan-1-ol
N-[(2R,3R)-1'-[(3-ethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide