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N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-4-oxo-4H-chromene-3-carboxamide
1-[benzyl(methyl)amino]-3-[4-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
1-(4-fluorophenyl)-4-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}butane-1,4-dione
2-(3-methylphenyl)-N-(1-{3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
4-chloro-1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)pyrrolidin-3-amine
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-3-methoxy-N-(oxolan-2-ylmethyl)benzamide
(4aR,7aS)-1-(2-ethylbutanoyl)-4-(furan-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-8-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-propyl-1H-1,2,3-triazol-4-yl)thiomorpholine-4-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)quinoxaline-6-carboxamide
2-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
4-(dimethyl-1,3-thiazole-5-carbonyl)-1-(2-methylphenyl)piperazin-2-one
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
4-{5-[1-(benzenesulfonyl)cyclopropyl]-3-methyl-1H-1,2,4-triazol-1-yl}-2-methylpyridine
{[2-(furan-2-yl)phenyl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-methyl-N-{1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-{[methyl(propan-2-yl)carbamoyl]methyl}-3-propylpiperidine-3-carboxylic acid
2-[1-({1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-[3-(difluoromethoxy)phenyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(3R,4S)-1-(2-hydroxy-4-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(3R,4R)-3-cyclopropyl-4-methyl-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-ol
2-{2,8-diazaspiro[4.5]decan-2-yl}-5-fluoro-N-methylpyrimidin-4-amine
(1R,3S)-7-(dimethyl-1,3-thiazole-5-carbonyl)-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
ethyl 1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-cyclopropyl-1-[1-(4-methylpyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(3E)-2-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}hept-3-enoic acid
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-4-yl)propan-1-one
1-[2-methoxy-4-({[2-(2-methoxyphenyl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-{2-[4-(2-fluorophenoxy)piperidin-1-yl]ethyl}-1H-indazole
3-(2-oxo-2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}ethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
1-(4,6-dimethylquinazolin-2-yl)-N-[2-(3-fluorophenyl)ethyl]piperidine-4-carboxamide
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
1-benzyl-8-(3-methylbutyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
6-fluoro-2-[({imidazo[1,2-a]pyridin-2-ylmethyl}amino)methyl]quinolin-4-ol
3-[3-(azocan-1-yl)propanamido]heptanoic acid
N-{4-[4-(thiomorpholin-4-yl)piperidin-1-yl]phenyl}cyclopentanecarboxamide
N-[(2R,3R)-2-methoxy-1'-(1-methyl-1H-indole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
N-methyl-3-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}pyridin-2-amine
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
N-[(5-chlorothiophen-2-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(1S,5R)-6-[3-(4-fluorophenoxy)propyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-(2-hydroxyethyl)-1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]methanesulfonamide
N,N-dimethyl-2-[2-(8-methylquinolin-5-yl)-1H-imidazol-1-yl]ethane-1-sulfonamide
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-1-[(3-methylquinoxalin-2-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(4-fluorophenyl)-4-[1-(3-methylbenzoyl)piperidin-3-yl]piperazine