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2-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}pyridine-3-carboxylic acid
5-benzyl-1-(4-methylphenyl)-4-propanoylpiperazin-2-one
(2R,3R,6R)-5-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-ethyl-2-[4-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)piperazin-1-yl]acetamide
2-amino-6-(2,2-dimethyloxan-4-yl)-4-[2-(2-hydroxyethoxy)phenyl]-5-methylpyridine-3-carbonitrile
8-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(4-methylpiperazin-1-yl)propanamide
(2S,4S)-4-amino-1-({2-[2-(4-methylpiperidin-1-yl)-2-oxoethoxy]phenyl}methyl)pyrrolidine-2-carboxylic acid
7-cyclohexyl-2-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
7-cyclohexyl-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(2-fluorophenyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-pyrazole-5-carboxamide
1-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-(2H-1,3-benzodioxol-5-yl)-3-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}urea
N-[(4-methoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
2-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(pyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
N-[(3-chlorophenyl)methyl]-N-propylpyridazine-3-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-(1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
7-(5-chloropyridin-2-yl)-4-(morpholine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
8-[5-(hydroxymethyl)furan-2-carbonyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(3-ethoxypropyl)amine
N,2-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
5-(2-{2-[(5,6-dimethylpyrimidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-(cyclopropylmethyl)-5-[2-(methylsulfanyl)benzoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3,5-difluoropyridine-2-carbonyl)-3-phenylpyrrolidin-3-ol
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(2-ethoxyphenyl)methyl]-N-ethylacetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,3-thiazole-5-carboxamide
methyl 5-{3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
1-cyclopropyl-3-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
3-{1-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-N-methylformamido}-N-methylbutanamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]propanamide
N-{2-[(2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)sulfanyl]phenyl}acetamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[(3-methoxyphenyl)amino]butanamide
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-thiazole-4-carboxamide
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
8-{[5-(hydroxymethyl)furan-2-yl]methyl}-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-({1-[1-(3,3-dimethylbutyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azepane
1-(1H-1,2,3-benzotriazol-5-yl)-3-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]urea
1-(5-methoxyfuran-2-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[1-(3-chlorobenzenesulfonyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
2-[1-(furan-3-ylmethyl)-4-[4-(pyridin-2-yl)pyrimidin-2-yl]piperazin-2-yl]ethan-1-ol
2-ethyl-4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholine