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ethyl 5-(2-chloro-6-fluorobenzoyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methyl-4-propyl-6-(1H-pyrazol-3-yl)pyrimidine
8-(cyclopentylmethyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxylate
5-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzothiadiazole
2-(2-methoxyethyl)-N-[3-(methylsulfanyl)propyl]-1,3-benzoxazole-6-carboxamide
(2S,4R)-N,N-diethyl-1-(furan-3-ylmethyl)-4-(2-methylfuran-3-amido)pyrrolidine-2-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
3-oxo-2-(prop-2-en-1-yl)-N-(thiophen-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{[(3-methylphenyl)methyl]amino}pyridine-3-carboxamide
2-(3-hydroxypropyl)-9-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N'-(2-fluoro-5-methylphenyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}butanediamide
2-[(4-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}piperidin-1-yl)methyl]pyridine
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
3-(3-methoxypropyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylic acid
1-[5-(2,2-diethylcyclopropanecarbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
N-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
4-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
7-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
4-(benzyloxy)-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-phenoxypropan-2-ol
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-(4-acetylpiperazin-1-yl)-3-(2-chlorophenyl)-3-phenylpropan-1-one
1-(4-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
N-[(2R,3R)-2-ethoxy-1'-[2-(phenylsulfanyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-phenoxypiperidine-4-carboxylic acid
(1S,5R)-3-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,5R,9R)-11-(2,5-dimethylbenzenesulfonyl)-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-[(8-{[3-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
4-({5-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-(3-fluorophenoxymethyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
N-[1-(furan-2-carbonyl)piperidin-3-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
1-{2-[(4-methylpiperidin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-[7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
1-({[3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-(2-methylphenyl)-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,4-diazepane
1-[3-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)phenyl]ethan-1-one
2-[4-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-(4-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}thiophen-2-yl)ethan-1-one
7-methyl-2-(4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
8-[(3-chloro-4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-3-(trifluoromethyl)pyridin-2-amine