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(1S,5R)-3-[4-(2-oxopyrrolidin-1-yl)butanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{6-carboxy-5-methylthieno[2,3-d]pyrimidin-4-yl}piperazine-2-carboxylic acid
(1R,2R,4R)-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
6-(1H-indol-3-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(ethylamino)-N-{[1-(methoxymethyl)cyclopentyl]methyl}pyrimidine-5-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-(isoquinoline-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-aminoethyl)-N-[1-(3-methylphenyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyridine-2-carboxamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3,5-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-indole-2-carboxamide
8-(4-methyl-1H-imidazole-5-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-ethyl-1-methyl-5-(2-methylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-7-yl]-2-methoxybenzamide
2-(2,1-benzoxazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
(2R,3R,6R)-3-(4-fluorophenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-1H-indol-3-yl)methyl]piperidin-3-amine
1-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]urea
3-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}pyridin-2-amine
1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]piperidine-4-carboxamide
3-[5-(2,3-dihydro-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
4-methyl-2-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
4-phenyl-N-{[1-(thiophen-3-ylmethyl)piperidin-3-yl]methyl}benzamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
2-methoxy-3-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}quinoline
N-{5-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]pyridin-2-yl}methanesulfonamide
2-methoxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
4-[(2-ethyl-1H-imidazol-1-yl)methyl]-2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazole
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(methylamino)ethan-1-one
N-(3-ethoxy-2-hydroxypropyl)-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(1,2-oxazol-3-ylmethyl)acetamide
2-(cyclohex-1-en-1-yl)-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-phenyl-3-[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrrolidine
1-cyclobutanecarbonyl-2-(4-fluorophenyl)piperidine
N,7-dimethyl-N-[1-(pyridin-3-yl)pentyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-(1-benzylpiperidin-4-yl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-cyclohexyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
5-methoxy-N-(1-methylpiperidin-4-yl)-4-oxo-N-(2-phenylethyl)-4H-pyran-2-carboxamide
5-fluoro-N-[1-(2-methoxyphenoxy)propan-2-yl]-1-methyl-1H-indole-2-carboxamide
N-ethyl-2-(4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)acetamide
{2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]ethyl}urea
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-N,4-dimethylpiperidine-4-carboxamide
(3S)-1-(5-{[(4,6-dimethylpyrimidin-2-yl)sulfanyl]methyl}furan-2-carbonyl)-N,N-dimethylazepan-3-amine
4-(2-{[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]oxy}hex-5-en-1-yl)-1,4-oxazepane
N-[(2S)-1-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-1-oxopropan-2-yl]acetamide
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-{[(pyridin-2-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
2-[4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)morpholin-3-yl]acetic acid
1-(2-ethoxyethyl)-2-oxo-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
8-methoxy-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide