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N-cyclooctyl-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{[(3-acetamidophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
N-methyl-4-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-4-oxobutanamide
3-(3-fluoro-4-methoxybenzoyl)-1-(thiophene-2-carbonyl)piperidine
1-tert-butyl-4-{[(7-methoxy-4-methylquinazolin-2-yl)(methyl)amino]methyl}pyrrolidin-2-one
2-[3-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenyl]-3,4,5,6,7,8-hexahydroquinazolin-4-one
(1R,3S,5S)-8-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
(4S)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-3,3,4-trimethylpiperidin-4-ol
4-(2,2-dimethylpropyl)-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
N-(2-methoxyethyl)-3-({1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}oxy)benzamide
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(4-chlorophenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}oxane-4-carboxamide
2-[(dimethylamino)methyl]-4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenol
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-{4-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]phenyl}acetamide
1-(2-methyl-5-propylpyrimidin-4-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]piperidin-4-amine
1-[4-(piperidine-1-carbonyl)pyridin-2-yl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N,N-dimethyl-N'-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)butanediamide
2-[3-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)-1H-indol-1-yl]acetamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2,6-dichloro-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}naphthalene-1-carboxamide
2-(2-{[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
5-({7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)-2-methoxyphenol
4-methyl-3-[(2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetamido)methyl]benzoic acid
N,2-dimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(5-methyl-1H-imidazol-4-yl)methyl]benzamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
[4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]methanol
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(pyridin-4-yl)ethyl]benzamide
N6-benzyl-N5-ethyl-N5-[2-(1H-pyrazol-1-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
6-{2-[5-(4-fluoro-2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrimidin-4-ol
N-cyclopropyl-3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}propanamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(5-chlorothiophen-2-yl)methyl]-3-methoxybenzamide
6-{[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
[2-(cyclohex-1-en-1-yl)ethyl]({[6-(4-ethylpiperazin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
N-[(3R,4S)-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
4-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-5-phenyl-2-(trifluoromethyl)pyrimidine
3-[(3-chlorophenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(3-hydroxybutyl)-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-1-methylazepane-2-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
(3S,7S)-5-(3-hydroxy-4-methoxybenzoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
(3S,4S)-1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol