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1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(4-methylphenyl)propan-1-one
5-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
1-(3-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
2-{[methyl(propan-2-yl)amino]methyl}-4-(pyrazin-2-yl)phenol
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-[2-(pyridin-4-yl)ethyl]imidazolidine-2,4-dione
N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
(3aR,5S,6S,7aS)-2-[(2-aminopyridin-3-yl)methyl]-octahydro-1H-isoindole-5,6-diol
2-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-6-(piperidin-4-yl)pyrimidin-4-amine
2-[(3-methoxyphenyl)methyl]-4-(1-propylpiperidin-4-yl)morpholine
1-[3-(morpholin-4-yl)propyl]-N-(1,2-oxazol-3-ylmethyl)-6-oxopiperidine-3-carboxamide
{3-[(1-methyl-1H-indol-5-yl)methyl]-9-propyl-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-(1-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N,3,5-trimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-benzofuran-2-carboxamide
1-methyl-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(2-cyclopentylacetyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-[3-(piperazine-1-sulfonyl)benzoyl]-1-oxa-7-azaspiro[3.5]nonane
N,4-dimethyl-5-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-amine
N-cyclohexyl-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[2-methyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]-4-oxobutanamide
2-amino-4-(6-ethoxypyridin-3-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
N-{1-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-methoxypropanamide
N-(1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}cyclopentyl)-4-methoxyaniline
5-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
2-chloro-4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methoxyphenol
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
1-methyl-4-{[3-(pyridin-2-yl)phenyl]methyl}piperazine-2-carboxylic acid
N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(3-methylpyridin-2-yl)piperazine-1-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[3-(pyrazin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-[1-(butane-1-sulfonyl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-6-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}phenol
8-(furan-2-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(3R,4S)-3-(2-carboxyethyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]benzoic acid
N-[1-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
2-(4-fluorophenyl)-N-[2-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
(1S,5R)-3-[(2,5-dimethylphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-[(2,3-dimethoxyphenyl)methyl]-2-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
N-methyl-N-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}thian-4-amine
9-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-hydroxy-2-(methylamino)propanamide
methyl 3-(6-methylpyridine-3-carbonyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-oxo-2-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)pyrrolidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
6-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1H-indole
7-(5-chloropyridin-2-yl)-9-methoxy-4-(2-methoxybenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine