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N2,N2-dimethyl-N4-[(3-phenyl-1H-pyrazol-5-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[(2R,3R)-2-methoxy-1'-(2-methylpropyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
ethyl 5-(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)-1H-imidazole-4-carboxylate
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4H-thieno[3,2-b]pyrrole-5-carboxamide
1-(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(N-methylmethanesulfonamido)propanamide
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-4-(4-fluorophenyl)-4-oxobutanamide
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-4-(trifluoromethyl)benzene-1-sulfonamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(trifluoromethyl)benzamide
N-({7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
1-benzyl-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylpropyl)amine
ethyl 4-(cyclopropylmethyl)-1-[(4-acetamidophenyl)methyl]piperidine-4-carboxylate
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
4-ethyl-1-[(4-methanesulfonylphenyl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}phenyl)amino]acetic acid
4-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-N,N-diethylaniline
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)(1,3-thiazol-2-ylmethyl)amine
(2S,4S)-4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
6-(2-methoxyphenyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
(1R,2S)-N-(prop-2-en-1-yl)-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]cyclohexane-1-carboxamide
3-[3-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-indazole
(2S,4R)-N-methyl-4-[(2-methyl-6-propylpyrimidin-4-yl)amino]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
methyl (2S,4R)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(3,4-difluorophenyl)methyl]pyrrolidine-2-carboxylate
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
ethyl({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(2-methylprop-2-en-1-yl)amine
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-2,6-dimethylpyridine-4-carboxamide
3-cyclohexyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
ethyl 4-({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)piperidine-1-carboxylate
(2E)-1-{4-[5-(3-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]pyrimidin-4-yl]piperidin-1-yl}-3-(pyridin-2-yl)prop-2-en-1-one
{5-[1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-imidazol-2-yl]furan-2-yl}methanol
3-(4-methoxyphenyl)-1-(1,2-oxazinan-2-yl)-3-phenylpropan-1-one
N-[2-(adamantan-1-yl)propan-2-yl]-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-(adamantan-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
1-(2-methoxyethyl)-8-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2S,4R)-1-[(2-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
(4aR,7aS)-1-[3-(1H-pyrazol-1-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-acetyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}thiophene-3-carboxamide
methyl 2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-methyl-2-oxopiperazin-1-yl)acetate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1H-imidazol-2-yl)benzamide
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
N-[(4-methoxyphenyl)methyl]-5-methyl-N-propylpyrazine-2-carboxamide
1-ethyl-4-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}piperazine
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
(1R,5S,6R)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-(2-methoxyethyl)-5-methyl-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]piperazine