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3-methyl-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
[2-(2-methoxyphenyl)ethyl]({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
(1S,5R)-6-benzyl-3-[(5-ethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
8-{1H-pyrrolo[2,3-b]pyridin-6-yl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}furan-2-carboxamide
1-(4-{[(1-hydroxybutan-2-yl)(thiophen-2-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
N-[(2,4-dihydroxyphenyl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
3-[3-(diphenylmethyl)-4H-1,2,4-triazol-4-yl]pyridine
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3,5-dimethoxy-2-{[methyl(oxan-4-ylmethyl)amino]methyl}benzoic acid
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-benzylpiperazin-1-yl)-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]propan-1-one
(3S,7S)-5-(1-methyl-1H-pyrazole-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-cycloheptyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidine-3-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
5-(2-fluorophenyl)-N-[2-(pyridin-3-yloxy)propyl]-1,2,4-triazin-3-amine
4-(3-hydroxypropyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,7aR)-1-(2,5-dimethylfuran-3-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
3-methoxy-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
(4aR,8aS)-6-[(3-ethoxy-4-hydroxyphenyl)methyl]-1-[2-(2-fluorophenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
6-chloro-2-(oxolane-3-carbonyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
4-[2-(4-chlorophenyl)morpholin-4-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
(3R,4R)-4-(azepan-1-yl)-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
4-(3-chlorothiophene-2-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
3-(thiophene-2-carbonyl)-1-[2-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
3-(2,3-dihydro-1H-isoindol-2-yl)-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]propan-1-one
1-(1-methylpiperidin-4-yl)-4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
9-ethyl-1-methyl-4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methyl-6-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-3-yl)pyrimidin-4-ol
3-[methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})amino]-1-phenylpropan-1-ol
(1S,5R)-6-[(3,5-difluorophenyl)methyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(5-chloropyridin-2-yl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,6-dimethyl-4-oxo-4H-pyran-2-carboxamide
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
7,7-dimethyl-2-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-1-phenylpyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-yl)-2-(1-propyl-1H-imidazol-2-yl)-1H-imidazole
1-ethyl-3-methyl-4-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
1-[2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetyl]piperidine-4-carbonitrile
N-[2-(dimethylamino)ethyl]-N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-(4-{5-butyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)-1H-imidazole
1-benzyl-8-(3-phenylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-(quinolin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-2-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}propanamide