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1-[3-(2-chlorophenyl)propyl]-4-cyclopentylpiperazine
3-{3-[(4-benzylpiperidin-1-yl)methyl]phenoxymethyl}-1-(1,3-thiazole-5-carbonyl)piperidine
5-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzothiadiazole
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
methyl (2S,4S)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
methyl({[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}acetamide
6-fluoro-2-({[2-(pyrrolidine-1-sulfonyl)ethyl]amino}methyl)quinolin-4-ol
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1,3-thiazole-4-carboxamide
1-(1H-1,3-benzodiazol-2-ylmethyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-{4-[4-(methoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
3-(1H-1,2,4-triazol-1-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
N-({1-[(2-cyanophenyl)methyl]piperidin-4-yl}methyl)pyridazine-3-carboxamide
(3S,9aR)-8-[(3-methoxyphenyl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 5-[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
2-{2-[4-benzyl-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepan-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-benzyl-1-ethyl-5-(2-methoxyacetamido)-N-methyl-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-8-methoxyquinoline
1'-(3-chloro-4-fluorobenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(4-methyl-1,4-diazepan-1-yl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-(piperazin-1-yl)ethan-1-one
9-methoxy-3-(2-phenylpropyl)-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[6-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-[(2-fluorophenyl)methyl]-N-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
ethyl 1-[(4-methoxyphenyl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
5-acetamido-1-(2-methoxyethyl)-N-(naphthalen-1-ylmethyl)-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
[3-(3-phenylpropyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl]methanol
N-[3-(azepan-1-yl)propyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[2-(dimethylamino)ethyl]-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
3-(2-methoxybenzoyl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
9-(cyclopropylmethyl)-4-[(2-ethylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-cyclohexyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-benzoxazole-6-carboxamide
9-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[1-(hydroxymethyl)cyclopropyl]methyl}-1-[3-(3-methylphenyl)phenyl]urea
3-(4-methylphenyl)-N-[2-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
2-[2-(dimethylamino)ethyl]-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(4-chlorobenzenesulfonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
(4aR,7aS)-1-acetyl-4-(4-ethylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 4-[(4-methoxyphenyl)methyl]-1-(2-methylfuran-3-carbonyl)piperidine-4-carboxylate
7-(2-methylphenyl)-4-(pyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(3,5-dimethoxybenzoyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-cyclopentyl-4-{3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
7-[(3,4-difluorophenyl)methyl]-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
4-[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]-5-ethyl-6-methylpyrimidin-2-amine
ethyl (4aS,8aR)-6-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylate
(3R,5S)-5-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-3-ol