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1-[4-(2-methoxyphenyl)phenyl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-[2-(propan-2-yloxy)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-1-methyl-6-oxo-N-(pyridin-3-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
6-methoxy-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-4-amine
1-benzyl-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
N1-(2-butyl-6-methylpyrimidin-4-yl)-N2-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}ethane-1,2-diamine
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](2-methylpropyl)(pyridin-2-ylmethyl)amine
5-[3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
N-[(2-fluoro-4-methoxyphenyl)methyl]-6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
2-(3-aminopyrrolidine-1-carbonyl)-6-(4-fluorophenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
6-ethyl-N-[2-hydroxy-3-(pyrrolidin-1-yl)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N2-[1-(4-methanesulfonylphenyl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
N-butyl-3-methyl-N-(3-phenylprop-2-yn-1-yl)furan-2-carboxamide
(3aS,6aS)-2-(1H-imidazol-4-ylmethyl)-5-(quinoxaline-6-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
2-{5-[(1R,9aR)-octahydro-1H-quinolizin-1-yl]-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl}acetamide
N-(3-hydroxypropyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)acetamide
1-ethyl-4-({3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrazole
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(thiophene-3-carbonyl)piperidin-3-yl]propan-1-ol
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(3-methyl-4-oxopentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-1H-indole
N-({3-methyl-7-[2-(methylsulfanyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-ethyl-5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]pyrimidine
N-[(2S,4R,6S)-2-ethyl-6-[1-(2-methoxyethyl)-1H-imidazol-2-yl]oxan-4-yl]benzamide
8-(5-chloropyridin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,3-oxazole-5-carboxamide
3-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}propane-1,2-diol
(2S,4S)-1-benzyl-N-ethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(1-methylcyclopropyl)benzamide
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2,2-dimethylpropan-1-one
3-(1-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1H-imidazol-2-yl)pyridine
N-cyclohexyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
2-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
N-methyl-2-(propan-2-yl)-N-(quinolin-2-ylmethyl)pyrimidine-4-carboxamide
(3S,4R)-1-(2-ethoxyethyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
5-benzyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
3-methyl-1-(2-methylpropyl)-4-[3-(pyridin-4-yl)propanoyl]piperazin-2-one
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-propyl-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
2-{4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}-7-fluoro-4,6-dimethylquinazoline
2-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1'-(1H-1,2,3-triazole-5-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
6-chloro-2-methyl-N-[2-(4-methylmorpholin-2-yl)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
(3S,4R)-4-phenyl-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]pyrrolidine-3-carboxylic acid
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[2-(4-fluorophenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
2-ethyl-5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]pyrimidine
methyl 3-[2-(4-fluorophenyl)acetyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3-methoxypropyl)(methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine