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N-[(2,6-difluoro-3-methoxyphenyl)methyl]-5-ethyl-1,3,4-oxadiazol-2-amine
(4aR,7aS)-1-methyl-4-[3-(2-methylphenyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-oxo-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
1-(3-ethynylbenzoyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
1-ethyl-N,5-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-3-carboxamide
1-benzyl-N3-[(2-benzyl-1,3-thiazol-4-yl)methyl]-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-2-yl)acetamide
1-cyclopropyl-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrrole-2-carboxamide
5-(2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[(4-ethylphenyl)methyl]-1-(1H-imidazol-1-ylmethyl)-N-(2-methoxyethyl)cyclopropane-1-carboxamide
4'-[(3,4-dimethoxypyridin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
N-(2-methylphenyl)-3-oxo-3-[3-(propoxymethyl)pyrrolidin-1-yl]propanamide
2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
[4-benzyl-1-(2,3-dimethoxybenzoyl)piperidin-4-yl]methanol
N-(cyclopropylmethyl)-2-[3-(2-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
[(3aS,6aS)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-4-carbonitrile
N-[(2-chlorophenyl)methyl]-5-(methoxymethyl)-N-(propan-2-yl)furan-2-carboxamide
N-({1-[(2,6-dimethylphenyl)methyl]piperidin-3-yl}methyl)pyrazine-2-carboxamide
1,5,6-trimethyl-2-oxo-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methylpyridine-3-carboxamide
ethyl 2-[2-({1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)ethyl]-1,3-thiazole-4-carboxylate
(3S,4S)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(propan-2-yloxy)pyrrolidin-3-ol
2-[2-methyl-3-({3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-indol-1-yl]acetamide
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
(1S,5R)-3-[(2-chloro-5-fluorophenyl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[methyl({4-methyl-5-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
4-{3-[3-(methylamino)propoxy]phenyl}benzoic acid
N-cyclopropyl-3-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}propanamide
N-(butan-2-yl)-4-methyl-N-[(4-methylphenyl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-(furan-2-ylmethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
N-{4-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]phenyl}cyclopentanecarboxamide
2-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-1,2-oxazinane
N-{[7-methoxy-2-(thiomorpholin-4-yl)quinolin-3-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
4,4,4-trifluoro-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]butan-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
(3S,4R)-4-methyl-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperidine-3,4-diol
(5S,9aS,9bS)-5-(2-chloro-4-fluorophenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{3-[2-(4-fluorophenyl)piperidine-1-carbonyl]phenoxy}acetamide
8-[(2-fluoro-5-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)phenoxy]acetamide
N-methyl-N-(pyridin-2-ylmethyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine