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N,N-dimethyl-5-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)pyrimidin-2-amine
1-benzyl-8-[(2,4-difluorophenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-1H-pyrazole-4-carboxamide
4-(8-chloro-2-methylquinoline-4-carbonyl)-3-(propan-2-yl)piperazin-2-one
3-cyclopropyl-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-1H-pyrazole-5-carboxamide
N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(1H-pyrazol-1-yl)benzamide
N-cyclopropyl-4-methoxy-3-{[1-(quinolin-8-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl 4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}benzoate
7-(propan-2-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1H-pyrazole-3-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2,5-dimethyl-N-(2-methylpropyl)furan-3-carboxamide
2-fluoro-N-[(8-{2-[4-(methylsulfanyl)phenyl]acetyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]benzamide
5-benzyl-5-[1-(2-ethylbutyl)piperidin-4-yl]-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
8-methoxy-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N,N-diethyl-1-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine-3-carboxamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[(1-methylpyrrolidin-3-yl)methyl]pyrimidin-2-amine
7-[(2,3-dimethoxyphenyl)methyl]-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-N-cyclopropylbenzamide
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}pyrrolidine-2,5-dione
{4-[(2-chlorophenyl)methyl]-1-(4-methoxybenzenesulfonyl)piperidin-4-yl}methanol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-(3,4-difluorophenyl)piperidine-1-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]acetamide
N,5-dimethyl-3-phenyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-4-carboxamide
methyl 3-benzyl-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{2-[(2-methoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
3-(1H-indol-3-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}propanamide
methyl 2-[8-(cyclohexylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(6-cyanopyridin-2-yl)piperidine-4-carboxylic acid
(2S,4S,5R)-4-[(carboxymethyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
2-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethane-1-sulfonamide
methyl 6-[2-(3-methylphenyl)acetyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-benzyl-4-[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]piperidine
4-({1-[4-(pyridin-2-yl)pyrimidin-2-yl]azetidin-3-yl}oxy)benzoic acid
1-(carbamoylmethyl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
6-methoxy-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}benzonitrile
7-(2-methylphenyl)-4-(5-propylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3-{2-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]pyrimidine-5-carboxamide
1-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[1-(pyrazin-2-yl)piperidin-3-yl]urea
4-(3-hydroxy-3-methylbutyl)-N-[1-(hydroxymethyl)cyclopentyl]benzamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
4-methyl-3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}benzene-1-sulfonamide
4-methyl-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-4-(1H-imidazol-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
methyl 4-(2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamido)butanoate
1-[2-(4H-1,2,4-triazol-4-ylmethyl)phenyl]-1H-1,2,4-triazole
methyl 3-[2-(cyclohex-1-en-1-yl)acetyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate