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N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)quinoline-8-sulfonamide
3-(4-methanesulfonylphenyl)-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
3-(5-methyl-1H-pyrazol-1-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
N-[(4-methoxyphenyl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)[(1-methyl-1H-indol-6-yl)methyl]amine
(5S,9aS,9bS)-2-cyclopentyl-5-(4-fluoro-3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-methyl-N-[1-(thian-4-yl)piperidin-4-yl]-1,3-benzothiazole-5-carboxamide
2-(4,5-dichloro-1H-imidazol-1-yl)-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
8-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
3-(cyclohex-3-ene-1-carbonyl)-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[(3-fluorophenyl)methyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
1-(4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-{5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1-methyl-1H-pyrazol-3-yl}-1,3,5-trimethyl-1H-pyrazole
6-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
methyl (2S,4S)-4-[3-(furan-2-amido)-2-methylbenzamido]-1-methylpyrrolidine-2-carboxylate
(4aR,8aS)-6-{[4-(methylsulfanyl)phenyl]methyl}-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-methyl-5-oxo-1-[4-(propan-2-yl)phenyl]-N-(thian-4-yl)pyrrolidine-3-carboxamide
1-[(1-hydroxycyclohexyl)methyl]-3-[3-(1H-imidazol-5-yl)phenyl]urea
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-1-ethyl-3-methylpiperazin-2-one
(5Z)-5-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethylidene]-1,3-thiazolidine-2,4-dione
N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2-chloro-6-fluorophenyl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)acetamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(1H-indol-3-ylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-({7-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzenesulfonamide
N-[3-(1H-imidazol-1-yl)butyl]-2,6,8-trimethylquinoline-4-carboxamide
1-methyl-1'-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(1S,5R)-6-(3-methyl-1H-pyrazole-5-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-[(2-methylpropyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-({1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
3-{1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-2-yl}propan-1-ol
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-6-methyl-2-propylpyrimidine
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}cyclopropanamine
3-(prop-2-en-1-yl)-1-[3-(thiophen-3-yl)propanoyl]piperidine-3-carboxylic acid
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3,4-dihydroquinazolin-4-one
4-{1-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]ethyl}morpholine
5-ethyl-5-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
N-[(3S,4R)-4-propyl-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(3-methoxypropyl)propanamide
N-{1-[7-(cyclopent-1-ene-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
N-[(2R,3R)-2-methoxy-1'-(1-methylcyclopropanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide