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N-[(4-fluorophenyl)methyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
3-(2-ethoxyethyl)-5-methyl-1-(2-phenylethyl)-1H-1,2,4-triazole
N-{[4-(cyclooctyloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
3-{1-[2-(4-chlorophenyl)acetyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
5-acetyl-N-(1-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-propylacetamide
(1R,5R)-6-benzyl-3-(3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(carbamoylamino)-N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}acetamide
N-[1-(3-methylpyridin-2-yl)propyl]pyrimidin-4-amine
2-(3,4-difluorophenyl)-N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-(3-fluoro-4-hydroxyphenyl)-1-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(3R,4R)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-3,4-dimethylpyrrolidin-3-ol
5-(2-chlorophenyl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-methylfuran-3-carboxamide
2-methyl-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-(1-{4-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]phenyl}-2,5-dimethyl-1H-pyrrol-3-yl)ethan-1-one
[(4-cyclopropyl-5-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(thiophen-2-ylmethyl)piperidine-3,5-dicarboxamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[1-(cyclohexylmethyl)piperidin-3-yl]acetamide
1-methyl-3-(2-phenylethyl)-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4S)-4-(propan-2-yl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-amine
4-benzyl-N-(5-chloro-2-methoxyphenyl)-4-(hydroxymethyl)piperidine-1-carboxamide
1-(2-methoxyethyl)-8-(2-phenylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3R,4S)-1-(3-fluorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
8-[2-(ethanesulfonyl)propanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
5-amino-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-phenyl-1H-pyrazole-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-4,4,4-trifluoro-N-(oxolan-2-ylmethyl)butanamide
5-[2-(2-chloro-4-fluorophenyl)acetyl]-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(3-methoxy-2-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(2R,3R)-2-methoxy-1'-(naphthalene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
5,6-dimethyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-2-carboxamide
5-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
{4-[1-(2-phenylethyl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
2-[4-(5-chloro-6-hydroxy-2-methylpyrimidin-4-yl)phenyl]-2-methylpropanenitrile
N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}cyclohexanecarboxamide
5-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-propyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
3-(2-cyclohexylacetyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{[4-(furan-2-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzoic acid
{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}[1-(1H-imidazol-1-yl)propan-2-yl]amine
(3-{5-[(pyridin-4-ylsulfanyl)methyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(phenylsulfanyl)ethan-1-one
1-[1-(3-hydroxy-2-methylbenzoyl)-4-phenylpiperidin-4-yl]ethan-1-one
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]propanamide