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2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
1-(2-chlorophenyl)-4-(3-hydroxybenzoyl)-5-methylpiperazin-2-one
1-(furan-2-ylmethyl)-4-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]piperidine
(4-{[1-(4-methylphthalazin-1-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
8-[(5-cyclopentylthiophen-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-chloro-N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-2-methylbenzene-1-sulfonamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(2-hydroxyphenyl)methyl]piperidine-4-carboxylate
1-benzyl-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-ethyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-amine
2-(4-methylphenoxy)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N,N-dimethylpyrrolidin-3-amine
N,N-dimethyl-6-(8-methylquinolin-5-yl)pyridine-3-carboxamide
2,7,8-trimethyl-4-[3-(trifluoromethyl)piperidine-1-carbonyl]quinoline
7-(2-methylbutyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
[(1-ethylpyrrolidin-3-yl)methyl](methyl){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-(adamantan-1-yl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]acetamide
1-[2-({1-[(4-chlorophenyl)methyl]piperidin-4-yl}amino)-4-methylpyrimidin-5-yl]ethan-1-one
(2S)-3-(2-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)propane-1,2-diol
3-(3-fluorophenyl)-3-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
5-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-{[3-(4-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]sulfonyl}pyrrolidine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
4-[(4-fluorophenyl)methyl]-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
3-(pyridin-4-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
ethyl 1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
1-[4-(quinolin-8-yl)phenyl]propan-2-one
(1S,5R)-3-[2-(1H-indazol-1-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-cyclopropanecarbonyl-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-ethoxy-4-methyl-2-{4-[(2,3,4-trimethoxyphenyl)methyl]-1,4-diazepan-1-yl}quinazoline
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(4-methyl-3-phenylpiperazin-1-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
methyl 5-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4,5-dimethyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
2-(3-methylbutyl)-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)-5-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-(cyclopropylmethyl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,4S)-1-(2-chloro-4-fluorobenzoyl)-4-(propan-2-yl)pyrrolidin-3-amine
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-4-(4-acetamido-1H-pyrazol-1-yl)benzamide
2,6-difluoro-4-methoxy-N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]benzamide
{[1-(4-methoxyphenyl)cyclopentyl]methyl}({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-methyl-N-(oxan-2-ylmethyl)-4-(piperidin-1-ylmethyl)benzamide
4-phenyl-3-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane
5-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-phenyl-1H-pyrazole
N-({7-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
N-(2,4-dimethylpentan-3-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide