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3-{2-[7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N-tert-butyl-4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidine-1-carboxamide
N-(2-{7-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-fluorobenzamide
N-(furan-3-ylmethyl)-4-{[(3R)-3-methylpiperazin-1-yl]sulfonyl}benzamide
4-[2-(adamantan-1-yl)acetyl]-3-(3-fluorophenyl)piperazin-2-one
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-[(5-methylpyrazin-2-yl)methyl]-8-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
2-(4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl)acetic acid
N-{[7-(2,6-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-cyclopentylpiperidine-3-carboxamide
1-(2,3-dihydro-1H-inden-4-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
4-(cyclobutylsulfamoyl)-N-[3-(methylsulfanyl)propyl]benzamide
N-(3,3-diphenylpropyl)-6-(1H-pyrazole-4-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropanecarboxamide
1-[4-(2-methoxyethyl)piperazin-1-yl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
1'-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[2-(2-methoxyphenyl)ethyl]-6-[(2,4,5-trimethylphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-({[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
2-methyl-N-[1-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
1-(3-methoxyphenyl)-4-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperazine
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[4-(1H-pyrazol-4-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
2-(oxolan-2-ylmethyl)-4-[4-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-{[(4-chlorophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
5-[6-(morpholine-4-carbonyl)pyrazin-2-yl]thiophene-2-carboxylic acid
5-(3-methoxyphenyl)-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]furan-2-carboxamide
1-(4-{[(dimethyl-1,2-oxazol-4-yl)methyl]amino}-2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-hydroxyethan-1-one
1-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-({8-cyclopropanecarbonyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(2,3,6-trifluorophenyl)acetamide
1-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
2-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(2-fluoro-5-methylphenoxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
1-(2-chlorobenzoyl)-3-(2-methoxybenzoyl)piperidine
1-[2-(dimethyl-1,3-thiazol-5-yl)ethyl]-4-(2-fluorophenoxy)piperidine
1-(5-acetyl-2-ethoxyphenyl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)urea
1-methyl-1'-[3-(piperazin-1-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(2-oxooxolan-3-yl)propanamide
N-[2-(3-methoxyphenyl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperidin-3-ol
(3aR,6aR)-N-[2-(ethanesulfonyl)ethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-methyl-2-[5-methyl-4-(pyrrolidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
1-cyclohexanecarbonyl-N-methyl-N-[4-(morpholin-4-yl)butyl]pyrrolidine-2-carboxamide
4-cyclopentyl-3-[3-(morpholin-4-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 4-(2-methoxyethyl)-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidine-4-carboxylate