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N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-cyclopropyl-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
2-(4-methoxyphenoxy)-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)benzamide
3-[(3-hydroxy-3-phenylpropyl)(methyl)amino]-N-(pyridin-3-yl)propanamide
methyl (2S,4R)-4-[3-(3-fluorophenyl)benzamido]-1-[(3-hydroxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
6-chloro-3-{[4-(6-ethoxy-4-methylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}-4H-chromen-4-one
5-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-propyl-1,2,4-oxadiazole
6-(1-benzothiophen-2-yl)-N-[2-(4-hydroxyphenyl)ethyl]-2-(morpholin-4-yl)pyridine-3-carboxamide
4-[(dimethylamino)methyl]-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]azepan-4-ol
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-4-ethylpiperazine
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pentanamide
N-[1-(pyridin-2-yl)propan-2-yl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
ethyl 4-({4-[2-(cyclohex-1-en-1-yl)acetyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate
2-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-2-azaspiro[4.4]nonan-3-one
4-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-hydroxybutyl)-1H-1,2,4-triazol-3-yl}benzamide
3-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-methylbenzamide
2,2-dimethyl-N-(1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidine
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(2-fluorophenyl)methyl]-5-methoxybenzamide
1-(4-methanesulfonylphenyl)-3-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}urea
6-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
2-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrazine
4-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-7-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2-hydroxy-2-phenylethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-fluoro-N-(1-{1-[4-(2-methylpropyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
4-(3-hydroxy-3-methylbutyl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)benzamide
4-{[3-({1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}morpholine
2-[3-(3-methoxybenzoyl)piperidin-1-yl]pyrimidin-4-amine
3-fluoro-4-(5-methylpyridin-3-yl)benzene-1-sulfonamide
N-cyclopropyl-1-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
6-(2-{[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]amino}ethyl)-2-methylpyrimidin-4-ol
1-[2-(1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
N-[2-(4-methylbenzenesulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
2-(1H-1,3-benzodiazol-2-ylmethyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
3-[2-(2,4-difluorophenyl)ethyl]-1-(1H-pyrrole-2-carbonyl)piperidine
3-[(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)methyl]-N,N-dimethylbenzamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(3-methylbutyl)propanamide
6-(2-hydroxyethyl)-N-[(2R)-1,1,1-trifluoro-3-methylbutan-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one