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methyl 3-(2,5-difluorobenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
N-cyclopentyl-5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[8-(2,3-difluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
4-(4-phenyl-1H-pyrazol-5-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
2-chloro-5-{4-[1-(morpholin-4-yl)ethyl]phenyl}benzoic acid
4-(cyclopropylmethyl)-1-[2-(ethylamino)pyrimidine-5-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
5-benzyl-5-{3-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-methyl-6-oxo-4-[(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
[(3R,4R)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
methyl 2-{[1-(4-methylquinazolin-2-yl)piperidin-4-yl]formamido}acetate
3-{[1-(2-hydroxyethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
5-(4-benzylpiperidine-1-carbonyl)-1-cyclopentyl-N,N-diethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(4-fluorophenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,3-oxazole-4-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-(4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazin-1-yl)-1,3-benzothiazole
4-{[({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]methyl}hepta-1,6-dien-4-ol
2,8-dimethyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
(7S,9aR)-N-benzyl-7-[(benzyloxy)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
5-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
(4aS,8aR)-1-(3-aminopropyl)-6-[(2-ethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[(5-chloro-1H-indol-2-yl)methyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-{[6-(5-aminopyridin-3-yl)pyrazin-2-yl]sulfanyl}acetic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
N-[(2R,3R)-1'-(dimethyl-1,2-oxazole-4-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
2-{[5-(1H-imidazol-1-ylmethyl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
5-methyl-3-(pyridin-4-ylmethyl)-5-{1-[2-(3,4,5-trimethoxyphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3aS,6aR)-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-{1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]ethyl}morpholine
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}-1,3-benzothiazole
1-{3-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-benzyl-8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-phenyl-5-(2,2,6,6-tetramethylpiperidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
3-[(3-fluorophenyl)methyl]-N-[2-(furan-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
3-ethyl-5-[(2S)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]-1,2,4-oxadiazole
5-(1,2-oxazinane-2-carbonyl)-2-(3-phenylpropyl)-1,3-benzoxazole
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(3-methoxypropyl)piperidine
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-methyl-1,8-naphthyridine-3-carboxamide
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-ethyl-4-oxo-N-(pyridin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
N-[(2R,3R)-2-methoxy-1'-(quinolin-8-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
9-(cyclopropylmethyl)-1-methyl-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-3-(2-phenylethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide