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5-benzyl-5-[1-(oxolane-2-carbonyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
4-(4-{[7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}phenyl)but-3-yn-1-ol
N-benzyl-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-N-methylpiperidin-3-amine
N-(1-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
1-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
2-butyl-4-(isoquinoline-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-methoxyquinoline-4-carbonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
2-{2-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}propan-1-one
methyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-(1-propylpiperidin-4-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-ethyl-2-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyridine
7-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
6-[3-fluoro-5-(2-methylpropoxy)phenyl]-N,N-dimethylpyridazin-3-amine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(3-fluorophenyl)-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
3-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-3-(2-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
1-(carbamoylmethyl)-N-[(dimethyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxamide
7-(3-hydroxy-2-methylbenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopropyl-3-[1-(furan-3-ylmethyl)piperidin-3-yl]propanamide
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2,3-dihydroxypropyl)acetamide
methyl 2-{[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)amino}acetate
3-(4-methylphenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}propan-1-one
methyl(2-phenoxyethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
methyl 2-{8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
(3S,4R)-1-(1-benzofuran-2-ylmethyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N4-cyclopropyl-6-(2,3,4-trimethoxyphenyl)pyrimidine-2,4-diamine
[(4aS,8aR)-6-[(2-chloro-5-methoxy-4-propoxyphenyl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
1-{4-[({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]phenyl}pyrrolidin-2-one
1-methyl-1-(1,2-oxazol-3-ylmethyl)-3-[5-(3-oxo-3-phenylpropyl)-1,3,4-thiadiazol-2-yl]urea
4-[1-(furan-3-ylmethyl)piperidin-3-yl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
5-(3-phenylpropyl)-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
1-cyclopentyl-N3,N3-diethyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
3-(1-benzyl-1H-imidazol-2-yl)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidine
{3-[(2,4-difluorophenyl)methyl]-1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl}methanol
N-[2-(2-chlorophenyl)ethyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
methyl N-{2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}carbamate
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-(2-oxoimidazolidin-1-yl)acetamide
3-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[(3R,4R)-1-[(4-fluoro-3-methylphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
2-[3-(2-amino-3-cyano-6-methyl-5,6,7,8-tetrahydroquinolin-4-yl)phenoxy]acetamide
1'-cyclopentyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(ethylsulfanyl)-5-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
2-(2H-1,3-benzodioxol-5-yloxy)-1-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}ethan-1-one