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2-(oxolan-2-ylmethyl)-4-(4-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,3,6-trimethyl-1-benzofuran-2-carboxamide
2-(2-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
methyl 4-[5-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
4-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzonitrile
5-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-(6-methoxypyrimidin-4-yl)piperazin-2-one
N,N-dimethyl-4-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperazine-1-carboxamide
2-chloro-4-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
7-(1-benzothiophen-3-yl)-9-ethoxy-4-(furan-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-(cyclopropylmethyl)-3-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-dimethyl-1-{[2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfonyl}pyrrolidin-3-amine
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
2-[(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2-phenylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(2-methoxyphenyl)methyl]piperazin-2-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-ol
2-methyl-4-(4-methylphenyl)-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-[4-(4-{[3-(dimethylamino)-2,2-dimethylpropyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
1-(3-chlorophenyl)-4-[1-(furan-3-ylmethyl)piperidin-3-yl]piperazine
N-[(4-fluorophenyl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-ethyl-4-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-1-(propan-2-yl)piperazine
N-cyclopropyl-4-({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)sulfamoyl)benzamide
8-methoxy-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(3-acetylphenoxymethyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,2R,6S,7S)-4-(2,3-dichlorobenzenesulfonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(3S,4S)-1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(naphthalen-2-yl)piperidin-3-ol
4-methoxy-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-(2-phenoxyethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(2R)-2-amino-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-methylpentanamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(2,2,6-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)propanamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]acetamide
2-[2-(2,2-diphenylethyl)morpholin-4-yl]propane-1,3-diol
7-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[({1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
ethyl 5-[(4-carbamoylpiperidin-1-yl)methyl]-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
1-{4-[(5-acetylthiophen-3-yl)methyl]-1,4-diazepan-1-yl}-2,2,2-trifluoroethan-1-one
3-[2-amino-4-(azetidin-1-yl)-6-methylpyrimidin-5-yl]propanoic acid
N,2,7-trimethyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[5-chloro-2-methoxy-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]acetic acid
(4aS,7aR)-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(3-chlorophenyl)-4-cyclobutanecarbonyl-9-(pyridin-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,5S)-N-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1,4-dithiepan-6-amine