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N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclohexanecarboxamide
1-methyl-3-{2-[3-(3-methylbutanoyl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
3-(4-fluorophenyl)-3-[(2-oxo-1,2-dihydroquinolin-4-yl)formamido]propanoic acid
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-(furan-3-ylmethyl)pyrrolidin-3-yl]cyclobutanecarboxamide
2-[3-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-2-carbonitrile
4-[(2-chlorophenyl)methyl]-1-cyclopentyl-1,4-diazepan-5-one
5-(dimethyl-1,3-thiazol-5-yl)isoquinoline
1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)acetamide
2-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
1-methyl-5-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
methyl 4-({1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)butanoate
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-{3-oxo-3-[2-(pyridin-2-yl)piperidin-1-yl]propyl}pyrrolidin-2-one
2-methyl-6-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-yl}pyrimidin-4-ol
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-ethyl-2-methylpyrimidine
{3-[(4-fluorophenyl)methyl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-yl}methanol
4-(4-ethoxy-3-methylphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}butanamide
2-[(3-methoxyphenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholine
2-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
2-(4-{4-[4-(2-methoxyphenoxy)piperidin-1-yl]piperidin-1-yl}phenyl)-1-(pyrrolidin-1-yl)ethan-1-one
(1S,4S)-2-(2-fluorophenyl)-5-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
N-ethyl-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-methyl-5-(3-methylphenyl)-4-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}pyrimidine
3-[1-(1-tert-butyl-5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]benzonitrile
N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2,7,8-trimethylquinoline-4-carboxamide
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
N-({1-[(3-chloropyridin-4-yl)methyl]pyrrolidin-3-yl}methyl)-2-hydroxypyridine-3-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-4-carboxylic acid
N-({7-[3-(dimethylamino)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]-3-(1H-1,2,3-benzotriazol-1-yl)propanamide
(3S,4S)-1-(3-methylbut-2-enoyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(2E)-2-methylbut-2-en-1-yl]amine
methyl 1-{[4-(1-methylcyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
(3R,4S)-4-(3-methoxyphenyl)-1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-amine
N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
4-[3-(cyclopropylmethyl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
(1S,5R)-3-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 4-{[(2-{5-oxo-1-[3-(pyridin-4-yl)propyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
4-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
5-acetyl-N-butyl-N-(furan-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3,5-dimethoxy-N-{[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}benzamide
(4aS,8aR)-6-(2-aminopyrimidin-4-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[({2-[2-(benzenesulfonyl)ethoxy]-7-chloroquinolin-3-yl}methyl)amino]ethan-1-ol