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(4aS,8aS)-2-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-decahydroisoquinolin-4a-ol
N-[2-(4-chlorophenyl)ethyl]-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-ethyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-4-carboxamide
N-[2-(diethylamino)ethyl]-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
(3R,4R)-1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(3-methoxyphenyl)methyl]piperazine
2-tert-butyl-6-(2-ethylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
methyl 2-(2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
4-(3-chloro-2-fluorophenyl)-5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-{3-[4-(morpholin-4-yl)butoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-(3,4-dimethylphenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-hydroxy-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}furan-2-carboxamide
N-[(2S,4R,6S)-2-(3-methyl-1H-pyrazol-5-yl)-6-(2-methylpropyl)oxan-4-yl]benzamide
3-[1-(3,5-dichloro-4-methylbenzoyl)piperidine-3-carbonyl]pyridine
(2S,4S)-4-amino-N,N-diethyl-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine-2-carboxamide
(3aR,6aR)-2-[(propan-2-yl)carbamoyl]-5-(pyridin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
8-fluoro-3-[2-(4-methylpiperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1H-indole
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-{3-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(4,6-dimethylpyrimidin-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-amine
N-[(2R,3R)-2-ethoxy-1'-{[2-(furan-2-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
[(2S)-1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)pyrrolidin-2-yl]methanol
2-(morpholin-4-yl)-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
N-ethyl-5-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine
1-[4-(8-methoxyquinolin-5-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
7-(2-hydroxyethyl)-2-[2-(2,3,6-trimethylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-({1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidin-4-yl}oxy)pyridine
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2,6-dimethoxybenzamide
3-{[1-(4-hydroxy-3-methoxybenzoyl)piperidin-4-yl]methyl}benzoic acid
3-(1H-1,3-benzodiazol-2-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
N-{[3-methyl-7-(2-phenoxypropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
7-(2-cyclohexylethyl)-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-benzyl-1-ethyl-N-[(6-methylpyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
8-(4-fluoro-2-methylbenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-aminoquinolin-8-yl)-N,N-bis(propan-2-yl)benzamide
3-(2-ethyl-1H-imidazol-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
N-[2-(dimethylsulfamoyl)ethyl]-2-methyl-1-benzofuran-5-carboxamide
1-(2-chlorophenyl)-4-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]piperazin-2-one
8-(4-methylbenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
N-cyclopropyl-3-ethoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(prop-2-en-1-yloxy)benzamide
1-(azocan-1-yl)-3-[5-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
dimethyl(3-{2-[1-(quinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
3-phenyl-N-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(3-ethoxy-2-hydroxypropyl)benzamide