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1-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}azepan-2-one
N-(2-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
1-[4-(methylamino)pyrimidin-2-yl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1,4-diazepane-6-carboxylic acid
N,N-dimethyl-2-({[3-(4H-1,2,4-triazol-4-yl)phenyl]formamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
7-fluoro-N-(morpholin-2-ylmethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-(quinolin-5-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
3-{5-[(2-chloro-6-fluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-[3-(4-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[(4,4-difluoropiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
{2,4,6-trimethyl-3-[({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)methyl]phenyl}methyl acetate
N-{2-[methyl(2-phenylethyl)amino]ethyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidine-3-carboxylate
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-methoxyethyl 2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
4-[2-(2-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-6-methoxyphenoxy)ethyl]morpholine
1-(2-methylfuran-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-(benzyloxy)-1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
6-methoxy-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-(3-methoxyphenoxymethyl)-N-(2,2,2-trifluoroethyl)-1H-pyrazole-3-carboxamide
N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]acetamide
N-[1-(adamantan-1-yl)propyl]-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-{2-[(cyclopentylamino)methyl]-5-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[(4-fluorophenyl)methyl]-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
methyl 2-[1-(3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-3-oxopiperazin-2-yl]acetate
2,6-dimethoxy-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
N-(pyridin-3-ylmethyl)-4-[6-(trifluoromethyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(2S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-amine
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-methylpropanamide
[(2R)-1-{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}pyrrolidin-2-yl]methanol
5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
2-amino-1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}ethan-1-one
5-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-amine
(3S,9aR)-3-(cyclohexylmethyl)-8-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4-{[1-(5-chloro-2-methoxybenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-(4-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[4-(propan-2-yloxy)phenyl]methyl}amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]pyrrolidin-3-yl]methanol
2-[(3-methoxyphenyl)methyl]-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]morpholine
1-(cyclopropylmethyl)-4-[(2E)-3-phenylprop-2-enoyl]-1,4-diazepane-6-carboxylic acid
2-methoxy-6-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)phenol
5,6-dimethoxy-2-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-1,2-dihydroisoquinolin-1-one
1-[2-(1,3-benzothiazol-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(2-phenylpropyl)piperidine-3-carboxamide
2-methoxy-1-{1'-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(5-{1-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
1-cyclohexyl-N-[(2-phenylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-[3-(3-chlorophenoxy)azetidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-(1-ethoxyethyl)-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(3-hydroxy-4-methylbenzoyl)piperidin-3-yl]pyrrolidin-2-one