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N-(1-methyl-1H-pyrazol-3-yl)-2-{2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}acetamide
3-[(3R,4S)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
4-[4-(2-ethylpiperidine-1-carbonyl)piperidin-1-yl]-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-methanesulfonyl-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
methyl 9-(benzyloxy)-3-[(2,3-dimethoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[3-(2-benzylmorpholin-4-yl)-3-oxopropyl]-2,3-dihydro-1H-isoindol-1-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
2-(4-methoxyphenyl)-N-{[1-(quinoline-6-carbonyl)piperidin-3-yl]methyl}acetamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-{1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-chlorophenyl)-4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}morpholine
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(2-methylphenyl)methyl]amino}methyl)piperidin-2-one
1-{6-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
1,9-dimethyl-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-6-methylpyridine-3-carboxylic acid
N,5-dimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-3-methylpiperidin-3-ol
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(1H-imidazol-1-yl)pyridazine
1-[2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)ethyl]-4-methylpiperazine
N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(4-methylphenyl)methyl]piperidine
(4S)-1-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-3,3,4-trimethylpiperidin-4-ol
3-(hydroxymethyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-ol
3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-N-(1,3-thiazol-2-yl)benzamide
2-(dimethylamino)-N-(3-methyl-1-{7-propanoyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
2-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
(2E)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-(1H-imidazol-4-yl)-N-(oxolan-2-ylmethyl)prop-2-enamide
5-[2-(benzylamino)ethyl]-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
3-ethyl-3-(oxolan-2-ylmethyl)-1-[4-(1H-pyrazol-4-yl)phenyl]urea
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-fluorophenyl)ethyl]propanamide
3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]-N-(1-propylpiperidin-4-yl)propanamide
N-[(2R,3R)-1'-(2,5-dimethylbenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{[4-(difluoromethoxy)phenyl]methyl}pyrrolidin-3-yl]methanol
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
2-[4-(3,5-dimethyl-1H-indole-2-carbonyl)-1-(furan-3-ylmethyl)piperazin-2-yl]ethan-1-ol
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
2-butyl-5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-1,3-benzoxazole
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(4-chlorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(4aR,8aS)-1-(2,2-diphenylethyl)-6-(pyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
(2S,4R)-4-amino-1-[2-(2,6-dichlorophenyl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-1,3-oxazole-4-carboxylate
5-(2-methoxy-4-methylphenoxymethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
2-{1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}quinoline
3-[(2S)-2,3-dihydroxypropyl]-1-(1-methyl-1H-indazol-5-yl)urea
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
5-chloro-4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
(2-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-2-yl}ethyl)dimethylamine
2-(adamantan-1-yl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylacetamide