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N-[(3,4-dimethoxyphenyl)methyl]-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(2-methylpropyl)piperidin-3-yl]propanamide
1-{8-butyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-[5-(2-methylpiperidine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]cyclobutanecarboxamide
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-(furan-2-ylmethyl)-N-methylacetamide
{3-[(3-methoxyphenyl)methyl]-1-(quinolin-2-ylmethyl)piperidin-3-yl}methanol
{3-[(2-methylphenyl)methyl]-1-(6-methylpyridine-2-carbonyl)piperidin-3-yl}methanol
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxylate
(2R,6R)-4-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(3S,4R)-1-(furan-2-ylmethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(2,4,5-trimethoxyphenyl)methyl]amine
methyl 2-{[1-(cyclohexylmethyl)-3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl](methyl)amino}acetate
9-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenyl)ethan-1-one
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-(pyridin-2-ylmethyl)piperidin-4-amine
4-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
7-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}-4-methyl-2H-chromen-2-one
N-({7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]furan-3-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-methoxy-2-methylpropyl)propanamide
3-(3-chlorophenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-phenylpropanamide
5-butyl-1'-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N,6-dimethyl-2-(piperidin-1-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-4-amine
2-{[3-(2-phenylethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
4-(3-hydroxy-3-methylbutyl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]benzamide
N-[(2-fluorophenyl)methyl]-3-[1-(thiophen-3-ylmethyl)piperidin-3-yl]propanamide
(4aS,7aR)-1-[(3-methoxyphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(4-chlorophenyl)cyclobutyl]-5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methoxyethoxy)ethan-1-one
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
N-benzyl[(1H-1,3-benzodiazol-5-yl)amino]sulfonamide
1-(1-benzothiophene-2-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
4-{2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}-1-(propan-2-yl)pyrrolidin-2-one
(2E)-4-methyl-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}pent-2-en-1-one
2-(3,4-dimethoxyphenyl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-{5-methyl-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-yl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-methyl-3-(thiomorpholine-4-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(5-methyl-1H-pyrazole-3-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(propan-2-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
2-[1-(cyclohexylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-[3-(pyrrolidin-1-yl)butyl]acetamide
N'-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-N,N-dimethylbutanediamide
N4-[(3-methoxy-2-propoxyphenyl)methyl]-5-methylpyrimidine-2,4-diamine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}acetic acid
3-(methoxymethyl)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
2-(5-{[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl)acetamide
6-methyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-[3-(difluoromethoxy)phenyl]pyridine-3-carbonitrile
1-(carbamoylmethyl)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)piperidine-4-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione