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1-methyl-2-oxo-8-{[4-(propan-2-yl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-ethyl-9-[2-(1H-imidazol-1-yl)acetyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-[2-({[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
N-[2-(2-chlorophenyl)ethyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
4-phenoxy-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
N-methyl-5-(1H-pyrazol-1-ylmethyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
2-[2-(furan-2-yl)pyrimidin-5-yl]-1-methyl-1H-1,3-benzodiazole
N-(2H-1,3-benzodioxol-5-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-amine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl)(1,3-thiazol-4-ylmethyl)amine
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-1-methyl-1H-pyrrole-2-carboxamide
3-{2-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
methyl 3-({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}carbamoyl)propanoate
N-[(2R,3R)-2-methoxy-1'-(3-phenylprop-2-yn-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
1-(1H-indole-2-carbonyl)-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(propan-2-yl)propanamide
9-[(3-chlorophenyl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-3-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-indole
1-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
(1R,2S)-N1-butyl-N2-[(5-methyl-1,2-oxazol-3-yl)methyl]cyclohexane-1,2-dicarboxamide
3-[5-(3,5-difluoropyridine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-(2-chlorophenyl)-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
5-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2R,3R)-2-methoxy-1'-(2,2,3,3-tetramethylcyclopropanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-[1-(1-cyclohexylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
6-[2-(hydroxymethyl)phenyl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
(2S,4R)-4-(4-{2-[(4-fluoro-3-methylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
4-[(2-fluorophenyl)methyl]-1-[4-(methylsulfanyl)benzoyl]-1,4-diazepan-5-one
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-indole
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
3-methyl-8-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
[(2S)-1-(4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidin-2-yl]methanol
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]propanamide
(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)piperidin-3-yl)methanol
4-({5-[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-pyrrole-2-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2,6-difluorobenzamide
(3-phenylprop-2-yn-1-yl)(propyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-(5-methyl-1,2-oxazol-3-yl)-2-[(2R)-oxolane-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-[4-(2-acetylbenzoyl)piperazin-1-yl]-2-[(2,3-dimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
6-[(6-methoxypyridin-3-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-(4-fluorophenyl)piperidin-3-amine
2-methoxy-5-{2-[4-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}pyridine
5-ethyl-6-methyl-N-[(5-methylpyrazin-2-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
N-[(5-ethylpyridin-2-yl)methyl]-N,4-dimethylpyrimidin-2-amine
1-methyl-4-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-diazepane
2,3-dimethyl-N-(1,2-oxazol-3-ylmethyl)quinoxaline-6-carboxamide