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4-[4-(3-acetylbenzoyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
2-(cyclopropylmethyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(pyridin-2-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)benzamide
(1R,5S)-8-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3,8-diazabicyclo[3.2.1]octane
1-[4-(difluoromethoxy)-2-methylphenyl]-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
2-({1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
N-(1-phenylethyl)-3-[4-(pyridin-4-yl)piperidin-1-yl]propanamide
(4aR,7aS)-1-propanoyl-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(furan-2-ylmethyl)(prop-2-en-1-yl){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
[(2-methoxyphenyl)methyl](propyl)(pyridin-2-ylmethyl)amine
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
N-{1-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]-2-(2,4-difluorophenyl)ethyl}-N-methylcyclopropanecarboxamide
3-cyclopropyl-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-butyl-4-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-oxo-1-phenylethyl)piperazine-2,3-dione
1-[(1S,5R)-6-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
5-(2-methylphenyl)-4-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-2-(pyridin-3-yl)pyrimidine
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-methyl-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]urea
3-(3-hydroxy-3-methylbutyl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-diethylacetamide
N-[(1-benzylpiperidin-4-yl)methyl]-3-(3-hydroxy-1,2-oxazol-5-yl)-N-methylpropanamide
N-[(2-methylphenyl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)-N-(prop-2-en-1-yl)propanamide
N-[4-({methyl[2-(1H-pyrazol-4-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
3-(2-methylphenyl)-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-ol
1-(2-chloro-3,5-difluorophenyl)-3-(5-oxo-1-propylpyrrolidin-3-yl)urea
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3,5-difluorophenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[(2R,3R)-1'-[(4-ethoxyphenyl)methyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
1-[(2-cyanophenyl)methyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
methyl[(6-methylpyridin-2-yl)methyl][1-(3-methylpyridin-2-yl)propan-2-yl]amine
1-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
1-cyclopentyl-3-(2-fluorophenyl)-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
N-(4-fluorophenyl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-amine
2-(2-methylpropyl)-6-{spiro[2.3]hexane-1-carbonyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-(3,4-dichlorophenyl)-1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-[(3-chlorophenyl)methyl]-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propanamide
4-(1H-pyrazol-1-yl)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
2-ethoxy-5-[2-({pyrazolo[1,5-a]pyridin-3-ylmethyl}amino)pyrimidin-4-yl]benzoic acid
methyl 8-(2H-1,3-benzodioxol-4-ylmethyl)-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methoxypropan-1-one
5-[3-(piperazin-1-yl)phenyl]-N-(propan-2-yl)thiophene-2-carboxamide
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{4-[(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)methyl]phenyl}-2-methylbutan-2-ol
2-(1H-1,3-benzodiazole-2-carbonyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-{[4-(morpholin-4-yl)phenyl]methyl}-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-3-benzyl-1-(4,6-dimethylpyrimidin-2-yl)-4-methylpiperidin-4-ol
(2S,4S)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(pyridin-2-ylsulfanyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide