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2-methoxy-1-{1'-[5-(propan-2-yl)pyrimidin-4-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-({[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
1-(benzyloxy)-8-[2-(2,4,6-trifluorophenyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
8-(4-methylbenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 2-{7-chloro-3-[(2-ethylpiperidin-1-yl)methyl]-2-oxo-1,2-dihydroquinolin-1-yl}acetate
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
(2S,4R)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
[(1R,3S,3aS,6aR)-3-(3-chloro-4-fluorophenyl)-1,5-diethyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
3-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
[(3-chloro-4-methoxyphenyl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-indole-2-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
5-methyl-3-(2-methyl-1H-imidazol-4-yl)-1H-indole
3-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-1-phenylpropan-1-ol
6-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}sulfonyl)-2,3-dihydro-1,3-benzoxazol-2-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
4-methanesulfonyl-2-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}morpholine
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
6-(cyclopropylmethoxy)-4-[2-(methylsulfanyl)benzoyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-{[5-(5-chloro-3-fluoropyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
methyl 3-[(phenylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazine-2-carboxylic acid
4-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-6-methyl-2-propylpyrimidine
7-(cyclobutylmethyl)-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
9-methoxy-3-[(4-methoxy-3-methylphenyl)methyl]-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(4-ethylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(1-hydroxy-2-methylpropan-2-yl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-{[4-(cyclooctyloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclopropanecarboxamide
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(2-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}phenoxy)acetic acid
3-(1-methoxypropyl)-4-[(2-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[4-(2-chloro-4-hydroxyphenyl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,6-dimethylpyrimidin-4-amine
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4,4,4-trifluorobutan-1-one
methyl 5-[(4-hydroxybutan-2-yl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-ethyl-5-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrimidine
3-(2H-1,3-benzodioxol-5-yl)-5-(thiophen-3-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propoxy]pyridine
N,1-bis(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-cyclopentyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-methoxy-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{4-[2-cyclobutyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2-(1H-imidazol-2-yl)benzamide
methyl[(3-{[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
6-chloro-N-(2-methoxyethyl)-2-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}quinazolin-4-amine
4-(4-{[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol