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N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(3R,4S)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclopentanecarboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-3-(2-chlorophenyl)-3-phenylpropanamide
ethyl 2-{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-2-yl}acetate
(2S)-N-[3-(1H-indol-2-yl)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-methyl-N'-phenyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)ethanediamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(3-methoxyphenyl)methyl]amine
2-methyl-4-{4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]phenyl}butan-2-ol
5-[2-(piperidin-1-yl)ethyl]-7-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-6-methyl-4H-pyran-4-one
2-amino-4-[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]-6-(5-methylpyridin-2-yl)pyridine-3-carbonitrile
4-fluoro-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
2-{4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
(3R,5R)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-methyl-4-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]pyridine
[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
4-ethyl-1-(naphthalen-1-ylmethyl)-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(4-methanesulfonylphenyl)methyl]azetidin-3-yl}-2-methylpiperidine
4-{[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenol
4-[1-(3,5-dimethoxybenzoyl)piperidin-3-yl]-5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidine
(4aS,8aR)-1-(2-phenylethyl)-6-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
1-[2-(pyridin-3-yloxy)phenyl]-3-[3-(pyrrolidin-1-yl)propyl]urea
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
(4S)-1-[(3-chloro-4-fluorophenyl)methyl]-3,3,4-trimethylpiperidin-4-ol
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(2S,4R)-4-amino-1-(2-{[5-(furan-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)-N-methylpyrrolidine-2-carboxamide
3-{[bis(2-hydroxyethyl)amino]methyl}-7-methyl-1,2-dihydroquinolin-2-one
5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4-propylpyrimidine
(3R)-1-({1-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}phenol
1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-3-[2-(5-methylfuran-2-yl)ethyl]urea
N-(3-chloro-4-propanamidophenyl)-2,3-dihydro-1-benzofuran-5-carboxamide
2-{3-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]phenyl}-5-methyl-1,3,4-thiadiazole
1-[(2,6-difluorophenyl)methyl]-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(diethylamino)-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
1-(4-chlorophenyl)-N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
N-{[7-(4-tert-butylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
N1,N1,N3-trimethyl-N3-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-1,3-dicarboxamide
1-[4-(dimethylamino)azepan-1-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
N-({7-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
1-methyl-2-oxo-8-(thiophene-2-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(2S)-N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-5-oxopyrrolidine-2-carboxamide
2-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(morpholine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
ethyl 4-[(2-chlorophenyl)methyl]-1-(3-phenylpropanoyl)piperidine-4-carboxylate
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea