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4-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-1-(propan-2-yl)piperidine
4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]-1-(3-hydroxyphenyl)pyrrolidin-2-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-6-ethyl-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-hydroxy-2,2-dimethylpropyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
3-methyl-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-4-(4-fluorophenyl)-4-oxo-N-(oxolan-2-ylmethyl)butanamide
1-cycloheptyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
methyl[(2-methyl-1H-imidazol-4-yl)methyl]{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
N-cyclopentyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-benzyl-N-(cyclobutylmethyl)-4-(pyrrolidin-3-yl)benzamide
3-[({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(prop-2-en-1-yl)amino]-1λ6-thiolane-1,1-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[2-(2-methoxyphenyl)ethyl]amino}piperidin-1-yl)benzamide
4-[(5-acetylthiophen-3-yl)methyl]-1λ6-thiomorpholine-1,1-dione
(1R,7S)-N-methyl-3-(3-methylbutyl)-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[4-(2-amino-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)-2-methoxyphenoxy]acetamide
4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-fluorophenyl)methyl]acetamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-[2-(1,3-thiazol-4-yl)acetyl]-1,4-diazepan-6-yl]oxy}acetamide
2,6-dimethoxy-N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}benzamide
1-[6-(cyclopropylmethoxy)-4-[(3-methoxyphenyl)methyl]-3-oxo-1,4-diazepan-1-yl]-4-phenylbutane-1,4-dione
1-cyclobutanecarbonyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide
5,7-dimethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-4,4,4-trifluorobutan-1-one
7-[(4-fluorophenyl)methyl]-N,N-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
3-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3,9-diazaspiro[5.5]undecane
1-[2-(pyridin-2-yl)-4-[(pyridin-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
1-methyl-4-{[5-(2-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}ethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
1-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
N-cyclohexyl-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}piperazin-2-one
8-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-pyrazol-1-yl)propanamide
2-(dimethyl-1,2-oxazol-4-yl)-1-(4-{2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)ethan-1-one
2-[4-(6-methyl-2-propylpyrimidin-4-yl)piperazin-1-yl]pyridine-3-carboxamide
2,7,8-trimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-4-carboxamide
4-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
3-chloro-N-[4-(4-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-one
N-(2-hydroxyethyl)-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-benzothiazole-5-carboxamide
4-{[2-(3,5-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}pyridine
2,2-dimethyl-N-(1-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
5-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
2-(2-methoxyethyl)-9-(pyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2H-1,3-benzodioxol-5-yl)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-(1-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-fluorobenzamide
4-[2-(pyrrolidin-1-yl)pyrimidine-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-[2-(4-methoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine-3-carboxamide
1-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]piperidin-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-phenylpropanamide