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2-[1-(3-fluorophenyl)-5-(3-oxo-1,2,3,4-tetrahydroquinoxalin-6-yl)-1H-1,2,4-triazol-3-yl]acetamide
(2S)-4-methyl-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-2-(propan-2-yl)piperazine
N-(3-cyano-4-methoxyphenyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-[1-(3,4-dimethoxybenzoyl)piperidin-4-yl]-2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazole
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(4-methyl-1H-imidazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-(1H-imidazol-1-ylmethyl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-ol
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetamide
3-methoxy-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-1-one
N-(2-methyl-1-{7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)propanamide
4-(2-cyclopropyl-4-hydroxypyrimidine-5-carbonyl)-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(oxan-2-ylmethyl)amine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(2R)-2-methylpiperazine-1-carbonyl]benzene-1-sulfonamide
1-cyclohexanecarbonyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5-phenyl-1,2,4-triazin-3-amine
1-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)ethan-1-one
4-ethyl-1-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2-(2-phenyl-1,3-thiazol-4-yl)-N-(pyridin-3-ylmethyl)acetamide
N-[2-(2-fluorophenoxy)ethyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(2R,6R)-4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-[4-(2-methoxyphenyl)piperazin-1-yl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-(1-methoxypropan-2-yl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
propyl 3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-cyclopropyl-3-(3,3-diphenylpiperidin-1-yl)propanamide
1-benzyl-4-(3,3,3-trifluoropropyl)-1,4-diazepan-6-ol
N-[(2,4-difluorophenyl)methyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
(3S,4R)-4-(3-fluorophenyl)-1-(4-sulfamoylbutanoyl)pyrrolidine-3-carboxylic acid
1-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)methyl]-1H-pyrazole
1,3-dimethyl-2,6-dioxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-phenyl-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-3-yl)propanamide
2-chloro-N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
ethyl 1-{2-[2,5-dioxo-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
3-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-5-fluorobenzonitrile
1-methyl-3-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-{[4-(dimethylamino)-1-ethylpiperidin-4-yl]methyl}pyrimidin-4-amine
N-[1-({methyl[(3-methyl-1H-indol-2-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
ethyl 2-{N-methyl-1-[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]formamido}acetate
4-ethyl-5-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidin-2-amine
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-(methoxymethyl)piperidine
N-[2-(ethylsulfanyl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(4-methylphenoxy)-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-4-carboxylic acid
1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carboxamide
1-[(2,4-difluorophenyl)methyl]-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}azepan-2-one
4-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1λ6-thiane-1,1-dione
N-(2-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(6-methylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(dimethyl-1,2-oxazol-4-yl)-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-(cyclohexylmethyl)-3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]piperazin-2-one